# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | JNJ-38877605 | SID137276033 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
2. | PX-866 | 4, PX-866 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
3. | TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
4. | Binimetinib | SID174006430 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
5. | TAK-285 | 34e, TAK-285 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
6. | GSK1059615 | GSK-1059615 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
7. | Decernotinib (VX-509) | DECERNOTINIB | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
8. | 6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | 14, ENMD-2076 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
9. | Voxtalisib (XL765) | VOXTALISIB | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
10. | Lapatinib | GW-572016 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
11. | AZD1152 | 5 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
12. | Barasertib (AZD1152-HQPA) | 34 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
13. | ALA1094408 | 49 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
14. | CP-724714 | 4 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
15. | CX-4945 (Silmitasertib) | 25n | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
16. | Pexidartinib | PEXIDARTINIB | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
17. | LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
18. | CYC116 | 13, CYC-116 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
19. | Gilteritinib | GILTERITINIB | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens | ||
20. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991900 | Inactive | nM | Homo sapiens |