# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ulixertinib (BVD-523) | ULIXERTINIB | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
2. | LGX 818 | ENCORAFENIB | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
3. | AZD1208 | 28 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
4. | ALA576982 | 7, AC220 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
5. | BAY 80-6946 (Copanlisib) | 46, BAY80-6946 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
6. | Capmatinib (INCB28060) | SID174006562 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
7. | Everolimus | EVEROLIMUS | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
8. | Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
9. | SU 14813 | SU-14813 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
10. | SNS-314 | SID103905586 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
11. | SAR407899 | 14C | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
12. | Hydroxyfasudil | hydroxyfasudil | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
13. | PF-04217903 | SID103905666 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
14. | Voxtalisib (XL765) | VOXTALISIB | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
15. | Baricitinib | BARICITINIB | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
16. | Motesanib | AMG-706 | Kd apparent | = | 3 | nM | ALA3991728 | 8.52 | Uncertain | nM | Homo sapiens | |
17. | ridaforolimus | RIDAFOROLIMUS | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
18. | LY2603618 | RABUSERTIB | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
19. | Ruxolitinib (INCB018424) | 3, INCB-018424 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens | ||
20. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991728 | Inactive | nM | Homo sapiens |