# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SGI 1027 | 4, SGI-1027 | Activity | 0 | ALA4836926 | Not Active | Homo sapiens | |||||
2. | ALA4780968 | PKUMDL-CLM-32; CLM-32 | EC50 | = | 29.1 | uM | ALA4678160 | 4.54 | nM | Homo sapiens | ||
3. | ALA4780968 | PKUMDL-CLM-32; CLM-32 | INH | 0 | ALA4678160 | Dose-dependent effect | % | Homo sapiens | ||||
4. | ALA4079762 | 28 | INH | 0 | ALA3992301 | Not Active | % | Homo sapiens | ||||
5. | ALA4105521 | 27 | INH | 0 | ALA3992301 | Not Active | % | Homo sapiens | ||||
6. | ALA4082223 | 25 | INH | 0 | ALA3992301 | Not Active | % | Homo sapiens | ||||
7. | ALA4081781 | 16 | INH | 0 | ALA3992301 | Not Active | % | Homo sapiens | ||||
8. | ALA4079762 | 28 | INH | 0 | ALA3992300 | Dose-dependent effect | % | Homo sapiens | ||||
9. | ALA4105521 | 27 | INH | 0 | ALA3992300 | Dose-dependent effect | % | Homo sapiens | ||||
10. | ALA4082223 | 25 | INH | 0 | ALA3992300 | Dose-dependent effect | % | Homo sapiens | ||||
11. | ALA4081781 | 16 | INH | 0 | ALA3992300 | Dose-dependent effect | % | Homo sapiens | ||||
12. | ALA443375 | 1, 10058-F4 | IC50 | = | 49 | uM | ALA3991966 | 4.31 | nM | Homo sapiens | ||
13. | ALA201467 | 2k | IC50 | = | 4.1 | uM | ALA3991966 | 5.39 | nM | Homo sapiens | ||
14. | ALA1958097 | 37R | IC50 | = | 51 | uM | ALA3991966 | 4.29 | nM | Homo sapiens | ||
15. | ALA255556 | 2e | IC50 | = | 23 | uM | ALA3991966 | 4.64 | nM | Homo sapiens | ||
16. | ALA490486 | 28RH | IC50 | = | 36 | uM | ALA3991966 | 4.44 | nM | Homo sapiens | ||
17. | ALA4066335 | 1RH-S-Me | IC50 | = | 18 | uM | ALA3991966 | 4.75 | nM | Homo sapiens | ||
18. | ALA4093899 | 1RH-NCN-1 | IC50 | = | 42 | uM | ALA3991966 | 4.38 | nM | Homo sapiens | ||
19. | ALA4086023 | #015 | IC50 | = | 6.5 | uM | ALA3991966 | 5.19 | nM | Homo sapiens | ||
20. | ALA4103943 | #474 | IC50 | = | 10 | uM | ALA3991966 | 5.00 | nM | Homo sapiens |