# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAY-091 | EUB0001564 | % inhibition | 16.22 | % | ALA4887779 | Not Active | % | Homo sapiens | |||
2. | ALA4580220 | EUB0000311 | % residual kinase activity | 94 | % | ALA4884529 | Not Active | % | Homo sapiens | |||
3. | BAY 293 | EUB0000320 | % residual kinase activity | 88 | % | ALA4881473 | Not Active | % | Homo sapiens | |||
4. | BAY-885 | BAY-885; 41 | % residual kinase activity | 100 | % | ALA4881291 | Not Active | % | Homo sapiens | |||
5. | ALA4860129 | 30 | IC50 | = | 1320 | nM | ALA4839364 | 5.88 | nM | Homo sapiens | ||
6. | ALA4850640 | 29 | IC50 | = | 907 | nM | ALA4839364 | 6.04 | nM | Homo sapiens | ||
7. | ALA4860779 | 28 | IC50 | = | 141 | nM | ALA4839364 | 6.85 | nM | Homo sapiens | ||
8. | ALA4875626 | 27 | IC50 | = | 270 | nM | ALA4839364 | 6.57 | nM | Homo sapiens | ||
9. | ALA4871998 | 26 | IC50 | = | 790 | nM | ALA4839364 | 6.10 | nM | Homo sapiens | ||
10. | BAY-8400 | 25; BAY-8400 | IC50 | = | 394 | nM | ALA4839364 | 6.41 | nM | Homo sapiens | ||
11. | ALA4849035 | 24 | IC50 | = | 551 | nM | ALA4839364 | 6.26 | nM | Homo sapiens | ||
12. | ALA4873263 | 23 | IC50 | = | 2160 | nM | ALA4839364 | 5.67 | nM | Homo sapiens | ||
13. | ALA4852502 | 22 | IC50 | = | 407 | nM | ALA4839364 | 6.39 | nM | Homo sapiens | ||
14. | ALA4868400 | 21 | IC50 | = | 314 | nM | ALA4839364 | 6.50 | nM | Homo sapiens | ||
15. | ALA4870563 | 20 | IC50 | = | 90 | nM | ALA4839364 | 7.05 | nM | Homo sapiens | ||
16. | ALA4869632 | 19 | IC50 | = | 197 | nM | ALA4839364 | 6.71 | nM | Homo sapiens | ||
17. | ALA4879247 | 18 | IC50 | > | 20000 | nM | ALA4839364 | nM | Homo sapiens | |||
18. | ALA4850455 | 17 | IC50 | = | 19700 | nM | ALA4839364 | 4.71 | nM | Homo sapiens | ||
19. | ALA4847559 | 16 | IC50 | > | 20000 | nM | ALA4839364 | nM | Homo sapiens | |||
20. | ALA4865476 | 15 | IC50 | = | 13000 | nM | ALA4839364 | 4.89 | nM | Homo sapiens |