| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  BAY-091 | EUB0001564 | % inhibition | 10.59 | % | ALA4888122 | Not Active | % | Homo sapiens | |||
| 2. |  BI 605906 | BI605906 | % Ctrl | 96 | % | ALA4887255 | Not Active | % | Homo sapiens | |||
| 3. |  ALA4580220 | EUB0000311 | % residual kinase activity | 106 | % | ALA4884257 | Not Active | % | Homo sapiens | |||
| 4. |  BAY-885 | BAY-885; 41 | % residual kinase activity | 100 | % | ALA4880995 | Not Active | % | Homo sapiens | |||
| 5. |  ALA4791586 | 39 | INH | 0 | ALA4737706 | Not Active | % | Homo sapiens | ||||
| 6. |  ALA4777349 | 38 | INH | 0 | ALA4737706 | Not Active | % | Homo sapiens | ||||
| 7. |  Staurosporine (DMSO solution) | 1 (Staurosporine) | IC50 | = | 6.63 | 10^-8M | ALA4720798 | 7.18 | nM | Homo sapiens | ||
| 8. |  ALA4750196 | 6g | Activity | = | 104.54 | % | ALA4720459 | % | Homo sapiens | |||
| 9. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405298 | % | Homo sapiens | |||
| 10. |  ALA4545456 | 24 | INH | = | 30.5 | % | ALA4387190 | % | Homo sapiens | |||
| 11. |  Abemaciclib | ABEMACICLIB | INH | = | 29 | % | ALA4387190 | % | Homo sapiens | |||
| 12. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379181 | nM | Homo sapiens | |||
| 13. |  ALA4459587 | DC-TEADin02 | INH | = | -5 | % | ALA4378933 | % | Homo sapiens | |||
| 14. |  CDK9-IN-7 | 21e | INH | = | 11 | % | ALA4377710 | % | Homo sapiens | |||
| 15. |  ALA4528675 | 8d-1 | INH | = | 9.02 | % | ALA4366325 | % | Homo sapiens | |||
| 16. |  ALA4574669 | (R,R)-36n | INH | 0 | ALA4351796 | Not Active | % | Homo sapiens | ||||
| 17. |  ALA4472294 | 11g | Activity | = | 94 | % | ALA4336841 | % | Homo sapiens | |||
| 18. |  ALA4568120 | G28_14 | Activity | = | 87 | % | ALA4335013 | % | Homo sapiens | |||
| 19. |  ALA4455512 | G3_9 | Activity | = | 57 | % | ALA4335013 | % | Homo sapiens | |||
| 20. | Staurosporine (DMSO solution) | 1 (Staurosporine) | IC50 | = | 5.11 | 10'-8M | ALA4328347 | 7.29 | nM | Homo sapiens |
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