# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (R)-(−)-Falcarinol | 20 | IC50 | = | 41.3 | uM | ALA4829570 | 4.38 | nM | Homo sapiens | ||
2. | ALA4874732 | (R)-2i | IC50 | = | 67.3 | uM | ALA4829570 | 4.17 | nM | Homo sapiens | ||
3. | (R)-(−)-Falcarinol | 20 | INH | = | 61.6 | % | ALA4829569 | % | Homo sapiens | |||
4. | ALA4874732 | (R)-2i | INH | = | 79.7 | % | ALA4829569 | % | Homo sapiens | |||
5. | (R)-(−)-Falcarinol | 20 | INH | = | 28.1 | % | ALA4829568 | % | Homo sapiens | |||
6. | ALA4874732 | (R)-2i | INH | = | 38.6 | % | ALA4829568 | % | Homo sapiens | |||
7. | (R)-(−)-Falcarinol | 20 | INH | = | 7.9 | % | ALA4829567 | % | Homo sapiens | |||
8. | ALA4874732 | (R)-2i | INH | = | 7.7 | % | ALA4829567 | % | Homo sapiens | |||
9. | (R)-(−)-Falcarinol | 20 | Activity | 0 | ALA4829566 | Active | Homo sapiens | |||||
10. | ALA4874732 | (R)-2i | Activity | 0 | ALA4829566 | Not Active | Homo sapiens | |||||
11. | Auglurant | 1 | IC50 | > | 100 | uM | ALA4039312 | nM | Homo sapiens | |||
12. | ALA5190568 | 48 | IC50 | > | 30 | uM | ALA5154401 | nM | Homo sapiens | |||
13. | ALA5180169 | 2g | INH | 0 | ALA5168664 | NA | % | Homo sapiens | ||||
14. | ALA1428 | 17a | IC50 | = | 29.8 | nM | ALA5168664 | 7.53 | nM | Homo sapiens |