# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5179617 | 10 | IC50 | = | 697 | nM | ALA5165846 | 6.16 | nM | Homo sapiens | ||
2. | ALA5207141 | 32k | IC50 | = | 42 | nM | ALA5139330 | 7.38 | nM | Homo sapiens | ||
3. | Dinaciclib (SCH727965) | DINACICLIB | IC50 | = | 0.007 | uM | ALA5136675 | 8.15 | nM | Homo sapiens | ||
4. | ALA5194833 | 27 | IC50 | = | 0.304 | uM | ALA5136675 | 6.52 | nM | Homo sapiens | ||
5. | ALA5169449 | 25 | IC50 | = | 0.029 | uM | ALA5136675 | 7.54 | nM | Homo sapiens | ||
6. | ALA5194202 | 24 | IC50 | = | 0.064 | uM | ALA5136675 | 7.19 | nM | Homo sapiens | ||
7. | ALA5187378 | 23 | IC50 | = | 0.05 | uM | ALA5136675 | 7.30 | nM | Homo sapiens | ||
8. | ALA5182767 | 18 | IC50 | = | 0.073 | uM | ALA5136675 | 7.14 | nM | Homo sapiens | ||
9. | ALA5191136 | 6 | IC50 | = | 0.156 | uM | ALA5136675 | 6.81 | nM | Homo sapiens | ||
10. | ALA5203891 | 4 | Kd | = | 27.3 | nM | ALA5126114 | 7.56 | nM | Homo sapiens | ||
11. | ALA4160662 | 2 | Kd | = | 16.2 | nM | ALA5126114 | 7.79 | nM | Homo sapiens | ||
12. | mevociclib | SY-1365 | IC50 | = | 20 | nM | ALA4408794 | 7.70 | nM | Homo sapiens | ||
13. | ALA4441405 | SY-314 | IC50 | = | 312 | nM | ALA4408794 | 6.51 | nM | Homo sapiens | ||
14. | ALA4436535 | SY-351 | IC50 | = | 367 | nM | ALA4408794 | 6.43 | nM | Homo sapiens | ||
15. | THZ1 | THZI | IC50 | = | 893 | nM | ALA4408784 | 6.05 | nM | Homo sapiens | ||
16. | THZ1 | THZI | IC50 | = | 371 | nM | ALA4408794 | 6.43 | nM | Homo sapiens | ||
17. | THZ531 | 3; THZ-531 | IC50 | = | 158 | nM | ALA4408794 | 6.80 | nM | Homo sapiens | ||
18. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379178 | nM | Homo sapiens | |||
19. | ALA4459587 | DC-TEADin02 | INH | = | 11 | % | ALA4378936 | % | Homo sapiens | |||
20. | CDK9-IN-7 | 21e | INH | = | 45 | % | ALA4377707 | % | Homo sapiens |