# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAY-091 | EUB0001564 | % inhibition | 10.3 | % | ALA4888123 | Not Active | % | Homo sapiens | |||
2. | ALA4580220 | EUB0000311 | % residual kinase activity | 85 | % | ALA4884256 | Not Active | % | Homo sapiens | |||
3. | BAY-885 | BAY-885; 41 | % residual kinase activity | 94 | % | ALA4880992 | Not Active | % | Homo sapiens | |||
4. | ALA4856177 | 37d | IC50 | = | 29.1 | nM | ALA4830405 | 7.54 | nM | Homo sapiens | ||
5. | ALA4753819 | BSJ-03-162; Exp 14 | IC50 | = | 857.2 | nM | ALA4828801 | 6.07 | nM | Homo sapiens | ||
6. | ALA4862284 | 22c | IC50 | = | 181 | nM | ALA4828801 | 6.74 | nM | Homo sapiens | ||
7. | ALA4862643 | 22b | IC50 | = | 155.1 | nM | ALA4828801 | 6.81 | nM | Homo sapiens | ||
8. | ALA4754873 | BSJ-01-175; Exp 2 | IC50 | = | 156 | nM | ALA4828801 | 6.81 | nM | Homo sapiens | ||
9. | ALA4872216 | 15h | IC50 | = | 293.2 | nM | ALA4828801 | 6.53 | nM | Homo sapiens | ||
10. | ALA4853964 | 15g | IC50 | = | 130.5 | nM | ALA4828801 | 6.88 | nM | Homo sapiens | ||
11. | ALA4853887 | 15f | IC50 | = | 87.6 | nM | ALA4828801 | 7.06 | nM | Homo sapiens | ||
12. | ALA4860981 | 15e | IC50 | = | 142.3 | nM | ALA4828801 | 6.85 | nM | Homo sapiens | ||
13. | ALA4866757 | 15d | IC50 | = | 67.6 | nM | ALA4828801 | 7.17 | nM | Homo sapiens | ||
14. | ALA4748005 | BSJ-02-108; Exp 10 | IC50 | = | 35.4 | nM | ALA4828801 | 7.45 | nM | Homo sapiens | ||
15. | ALA4864697 | 15b | IC50 | = | 93.6 | nM | ALA4828801 | 7.03 | nM | Homo sapiens | ||
16. | ALA4866812 | 15a | IC50 | = | 166.7 | nM | ALA4828801 | 6.78 | nM | Homo sapiens | ||
17. | ALA4758566 | BSJ-03-055; Exp 7 | IC50 | = | 231.7 | nM | ALA4828801 | 6.63 | nM | Homo sapiens | ||
18. | ALA4787545 | BSJ-01-202; Exp 4 | IC50 | = | 764.9 | nM | ALA4828801 | 6.12 | nM | Homo sapiens | ||
19. | ALA4870659 | 10f | IC50 | = | 1450 | nM | ALA4828801 | 5.84 | nM | Homo sapiens | ||
20. | ALA4861833 | 10e | IC50 | = | 68.7 | nM | ALA4828801 | 7.16 | nM | Homo sapiens |