# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tetraethylthiuram disulfide | disulfiram | IC50 | = | 14.6 | uM | ALA5231856 | 4.84 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
2. | ALA4475926 | 6 | Activity | 0 | ALA4393318 | Active | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||||
3. | ALA4475926 | 6 | INH | 0 | ALA4393317 | Active | % | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||||
4. | ALA4475926 | 6 | Ratio | = | 7 | ALA4393316 | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||||
5. | ALA11350 | 1 | Activity | 0 | ALA4393315 | Not Active | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||||
6. | ALA4475926 | 6 | Ki | = | 36.6 | uM | ALA4393314 | 4.44 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
7. | ALA11350 | 1 | Ki | = | 127 | uM | ALA4393314 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||
8. | 3,4-Dihydroxybenzaldehyde | 4 | Kd | = | 220 | uM | ALA4393313 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||
9. | ALA1595473 | SID24834861 | Kd | = | 7.6 | uM | ALA4393313 | 5.12 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
10. | ALA4475926 | 6 | Kd | = | 7.6 | uM | ALA4393313 | 5.12 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
11. | ALA1368663 | SID4258187 | Kd | = | 7.6 | uM | ALA4393313 | 5.12 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
12. | ESI-08 | 1, ESI-08 | Kd | = | 7.6 | uM | ALA4393313 | 5.12 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
13. | ALA4544405 | 3 | Kd | = | 7.6 | uM | ALA4393313 | 5.12 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
14. | ALA421 | 18 | Kd | = | 7.6 | uM | ALA4393313 | 5.12 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
15. | ALA11350 | 1 | Kd | = | 14.1 | uM | ALA4393313 | 4.85 | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
16. | 3,4-Dihydroxybenzaldehyde | 4 | Kdiss | = | 4.18 | 10'-2/s | ALA4393312 | 10'-2/s | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||
17. | ALA4475926 | 6 | Kdiss | = | 3 | 10'-2/s | ALA4393312 | 10'-2/s | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||
18. | 3,4-Dihydroxybenzaldehyde | 4 | Ka | = | 1.88 | 10'2/M/s | ALA4393311 | 10'2/M/s | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||
19. | ALA4475926 | 6 | Ka | = | 3.2 | 10'3/M/s | ALA4393311 | 10'3/M/s | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | |||
20. | ALA4475926 | 6 | INH | > | 50 | % | ALA4393310 | % | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) |