# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | LDC1267 | 7; LDC1267 | % of control | < | 10 | % | ALA5212934 | % | Homo sapiens | |||
2. | Acalabrutinib (ACP-196) | ACALABRUTINIB | IC50 | > | 10 | uM | ALA5213047 | nM | Homo sapiens | |||
3. | ALA4065365 | 6l; E738 | IC50 | = | 10.7 | nM | ALA5151636 | 7.97 | nM | Homo sapiens | ||
4. | ALA3238113 | 1, B9 | IC50 | = | 2.8 | uM | ALA5131876 | 5.55 | nM | Homo sapiens | ||
5. | ALA44577 | 2 | IC50 | < | 0.5 | nM | ALA5128208 | nM | Homo sapiens | |||
6. | LASW1393 | 34 | INH | < | 50 | % | ALA4416509 | % | Homo sapiens | |||
7. | Zanubrutinib (BGB-3111) | BDBM250082 | INH | 0 | ALA4414993 | Not Active | % | Homo sapiens | ||||
8. | ALA4445335 | Roxyl-ZV-5J | INH | = | 33 | % | ALA4408014 | % | Homo sapiens | |||
9. | ALA4445335 | Roxyl-ZV-5J | INH | = | 66 | % | ALA4408013 | % | Homo sapiens | |||
10. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405397 | % | Homo sapiens | |||
11. | ALA4559936 | (+/-)-6 | Activity | = | 100 | % | ALA4391370 | % | Homo sapiens | |||
12. | ALA4564973 | 50 | INH | = | 76 | % | ALA4389744 | % | Homo sapiens | |||
13. | ALA4555459 | 43 | INH | = | 98 | % | ALA4389267 | % | Homo sapiens | |||
14. | ALA4473365 | 7c | Activity | = | 49 | % | ALA4382548 | % | Homo sapiens | |||
15. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379350 | nM | Homo sapiens | |||
16. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379349 | nM | Homo sapiens | |||
17. | ALA4459587 | DC-TEADin02 | INH | = | 3 | % | ALA4378842 | % | Homo sapiens | |||
18. | ALA4459587 | DC-TEADin02 | INH | = | -12 | % | ALA4378843 | % | Homo sapiens | |||
19. | CDK9-IN-7 | 21e | INH | = | 5 | % | ALA4377882 | % | Homo sapiens | |||
20. | CDK9-IN-7 | 21e | INH | = | 9 | % | ALA4377881 | % | Homo sapiens |