# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5174202 | 1; JTP-59557 | IC50 | = | 120 | nM | ALA5157676 | 6.92 | nM | Homo sapiens | ||
2. | ALA5171732 | 3 | IC50 | = | 64 | nM | ALA5157658 | 7.19 | nM | Homo sapiens | ||
3. | ALA5172873 | 14 | IC50 | = | 83 | nM | ALA5157658 | 7.08 | nM | Homo sapiens | ||
4. | ALA5194399 | 13 | IC50 | = | 33 | nM | ALA5157658 | 7.48 | nM | Homo sapiens | ||
5. | ALA5208550 | 12 | IC50 | = | 315 | nM | ALA5157658 | 6.50 | nM | Homo sapiens | ||
6. | ALA5189512 | 11 | IC50 | = | 40 | nM | ALA5157658 | 7.40 | nM | Homo sapiens | ||
7. | ALA5174328 | 10 | IC50 | < | 100 | nM | ALA5157658 | nM | Homo sapiens | |||
8. | ALA5192802 | 9 | IC50 | < | 100 | nM | ALA5157658 | nM | Homo sapiens | |||
9. | ALA5188634 | 8 | IC50 | = | 997 | nM | ALA5157658 | 6.00 | nM | Homo sapiens | ||
10. | ALA5194891 | 7 | IC50 | = | 354 | nM | ALA5157658 | 6.45 | nM | Homo sapiens | ||
11. | ALA5203083 | 6 | IC50 | = | 249 | nM | ALA5157658 | 6.60 | nM | Homo sapiens | ||
12. | ALA5205017 | 5 | IC50 | = | 404 | nM | ALA5157658 | 6.39 | nM | Homo sapiens | ||
13. | ALA5198191 | 4 | IC50 | = | 455 | nM | ALA5157658 | 6.34 | nM | Homo sapiens | ||
14. | ALA5209124 | 3 | IC50 | = | 87 | nM | ALA5157658 | 7.06 | nM | Homo sapiens | ||
15. | ALA5174202 | 1; JTP-59557 | IC50 | = | 838 | nM | ALA5157658 | 6.08 | nM | Homo sapiens | ||
16. | ALA4286458 | 005.2HCl | pIC50 | 0 | ALA4257143 | Not Determined | Homo sapiens | |||||
17. | ALA4281361 | 004.2HCl | pIC50 | 0 | ALA4257143 | Not Determined | Homo sapiens | |||||
18. | ALA3901000 | 003 | pIC50 | 0 | ALA4257143 | Not Determined | Homo sapiens | |||||
19. | Tenapanor hydrochloride | TENAPANOR HYDROCHLORIDE | pIC50 | < | 4.5 | ALA4257143 | nM | Homo sapiens | ||||
20. | ALA4289255 | 3; 001 | pIC50 | 0 | ALA4257143 | Not Determined | Homo sapiens |