# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4848627 | TAT-JYX-3 | t1/2 | = | 1.53 | s | ALA4837027 | hr | Homo sapiens | |||
2. | ALA4850575 | JYX-3 | t1/2 | = | 1.52 | s | ALA4837027 | hr | Homo sapiens | |||
3. | ALA4848627 | TAT-JYX-3 | Kd | = | 0.8 | uM | ALA4837026 | 6.10 | nM | Homo sapiens | ||
4. | ALA4850575 | JYX-3 | Kd | = | 0.37 | uM | ALA4837026 | 6.43 | nM | Homo sapiens | ||
5. | ALA4848627 | TAT-JYX-3 | IC50 | = | 1.74 | uM | ALA4837025 | 5.76 | nM | Homo sapiens | ||
6. | ALA4850575 | JYX-3 | IC50 | = | 0.41 | uM | ALA4837025 | 6.39 | nM | Homo sapiens | ||
7. | ALA4859531 | 7 | Activity | 0 | ALA4810358 | Not Active | Homo sapiens | |||||
8. | ALA4865432 | 24 | INH | 0 | ALA4810346 | Active | % | Homo sapiens | ||||
9. | ALA4863719 | 11 | INH | 0 | ALA4810346 | Active | % | Homo sapiens | ||||
10. | ALA4859531 | 7 | INH | 0 | ALA4810346 | Active | % | Homo sapiens | ||||
11. | ALA4855926 | 1 | INH | 0 | ALA4810346 | Active | % | Homo sapiens | ||||
12. | ALA4865432 | 24 | IC50 | = | 729 | nM | ALA4810341 | 6.14 | nM | Homo sapiens | ||
13. | ALA4863719 | 11 | IC50 | = | 984 | nM | ALA4810341 | 6.01 | nM | Homo sapiens | ||
14. | ALA4859531 | 7 | IC50 | = | 4934 | nM | ALA4810341 | 5.31 | nM | Homo sapiens | ||
15. | ALA4855926 | 1 | IC50 | = | 1850 | nM | ALA4810341 | 5.73 | nM | Homo sapiens | ||
16. | ALA4206834 | 28 | Ki | = | 9 | nM | ALA4202266 | 8.05 | nM | Homo sapiens | ||
17. | ALA4211714 | 27 | Ki | = | 23 | nM | ALA4202266 | 7.64 | nM | Homo sapiens | ||
18. | ALA4211204 | 26 | Ki | = | 13 | nM | ALA4202266 | 7.89 | nM | Homo sapiens | ||
19. | ALA4216170 | 25 | Ki | = | 57 | nM | ALA4202266 | 7.24 | nM | Homo sapiens | ||
20. | ALA4216933 | 24 | Ki | = | 50 | nM | ALA4202266 | 7.30 | nM | Homo sapiens |