# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 5-[(4-Chlorophenyl)sulfanyl]-1,2,3- thiadiazole-4-carboxylic acid | CCPST | Ki | = | 4500 | nM | ALA4827644 | 5.35 | nM | Mus musculus | ||
2. | ALA4864519 | 7 | IC50 | = | 7.7 | nM | ALA4827637 | 8.11 | nM | Mus musculus | ||
3. | ALA4857427 | Cpd A | IC50 | = | 14.6 | nM | ALA4827637 | 7.84 | nM | Mus musculus | ||
4. | ALA2260704 | 9 | FC | = | 0.88 | ALA4234435 | Mus musculus | |||||
5. | ALA4247590 | 26 | Ratio EC50 | = | 7 | ALA4234448 | Mus musculus | |||||
6. | Calconcarboxylic acid | 2i | FC | = | 1.11 | ALA4234435 | Mus musculus | |||||
7. | ALA4237565 | 27 | Ratio EC50 | = | 7 | ALA4234448 | Mus musculus | |||||
8. | ALA4242089 | 55 | INH | = | 30 | % | ALA4234457 | % | Mus musculus | |||
9. | ALA4241120 | 54 | INH | = | 30 | % | ALA4234457 | % | Mus musculus | |||
10. | ALA4245056 | 31 | INH | = | 30 | % | ALA4234457 | % | Mus musculus | |||
11. | ALA4247590 | 26 | Ratio EC50 | = | 5 | ALA4234449 | Mus musculus | |||||
12. | ALA4237565 | 27 | INH | 0 | ALA4234446 | Active | % | Mus musculus | ||||
13. | ALA4237565 | 27 | INH | = | 26.5 | % | ALA4234445 | % | Mus musculus | |||
14. | ALA4237565 | 27 | EC50 | = | 9.2 | uM | ALA4234444 | 5.04 | nM | Mus musculus | ||
15. | ALA4247590 | 26 | EC50 | = | 11.19 | uM | ALA4234444 | 4.95 | nM | Mus musculus | ||
16. | ALA4237565 | 27 | EC50 | = | 7.88 | uM | ALA4234443 | 5.10 | nM | Mus musculus | ||
17. | ALA4247590 | 26 | EC50 | = | 8.36 | uM | ALA4234443 | 5.08 | nM | Mus musculus | ||
18. | ALA4237565 | 27 | EC50 | = | 3.59 | uM | ALA4234442 | 5.45 | nM | Mus musculus | ||
19. | ALA4247590 | 26 | EC50 | = | 3.45 | uM | ALA4234442 | 5.46 | nM | Mus musculus | ||
20. | ALA4247590 | 26 | INH | = | 62.3 | % | ALA4234440 | % | Mus musculus |