# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5179617 | 10 | IC50 | > | 1000 | nM | ALA5165847 | nM | Homo sapiens | |||
2. | Dinaciclib (SCH727965) | DINACICLIB | IC50 | = | 0.021 | uM | ALA5136676 | 7.68 | nM | Homo sapiens | ||
3. | ALA5194833 | 27 | IC50 | = | 0.334 | uM | ALA5136676 | 6.48 | nM | Homo sapiens | ||
4. | ALA5169449 | 25 | IC50 | = | 0.012 | uM | ALA5136676 | 7.92 | nM | Homo sapiens | ||
5. | ALA5194202 | 24 | IC50 | = | 0.022 | uM | ALA5136676 | 7.66 | nM | Homo sapiens | ||
6. | ALA5187378 | 23 | IC50 | = | 0.022 | uM | ALA5136676 | 7.66 | nM | Homo sapiens | ||
7. | ALA5182767 | 18 | IC50 | = | 0.067 | uM | ALA5136676 | 7.17 | nM | Homo sapiens | ||
8. | ALA5191136 | 6 | IC50 | = | 0.122 | uM | ALA5136676 | 6.91 | nM | Homo sapiens | ||
9. | ALA5203891 | 4 | Kd | = | 17 | nM | ALA5126115 | 7.77 | nM | Homo sapiens | ||
10. | ALA4160662 | 2 | Kd | = | 8.6 | nM | ALA5126115 | 8.07 | nM | Homo sapiens | ||
11. | THZ1 | THZI | IC50 | = | 628 | nM | ALA4408787 | 6.20 | nM | Homo sapiens | ||
12. | THZ531 | 3; THZ-531 | IC50 | = | 69 | nM | ALA4408795 | 7.16 | nM | Homo sapiens | ||
13. | ALA4545456 | 24 | INH | = | 50 | % | ALA4387186 | % | Homo sapiens | |||
14. | Abemaciclib | ABEMACICLIB | INH | = | 38 | % | ALA4387186 | % | Homo sapiens | |||
15. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379179 | nM | Homo sapiens | |||
16. | ALA4459587 | DC-TEADin02 | INH | = | 17 | % | ALA4378935 | % | Homo sapiens | |||
17. | CDK9-IN-7 | 21e | INH | = | 26 | % | ALA4377708 | % | Homo sapiens | |||
18. | THZ531 | 3; THZ-531 | IC50 | = | 69 | nM | ALA4775151 | 7.16 | nM | Homo sapiens | ||
19. | ALA4574669 | (R,R)-36n | INH | 0 | ALA4351792 | Not Active | % | Homo sapiens | ||||
20. | ALA4472294 | 11g | Activity | = | 84 | % | ALA4336837 | % | Homo sapiens |