| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  BAY-091 | EUB0001564 | % inhibition | 18.05 | % | ALA4888118 | Not Active | % | Homo sapiens | |||
| 2. |  BAY-885 | BAY-885; 41 | % residual kinase activity | 117 | % | ALA4880994 | Not Active | % | Homo sapiens | |||
| 3. |  ALA4434727 | 100, 101; FMF-04-159-2 | IC50 | = | 39.6 | nM | ALA4434185 | 7.40 | nM | Homo sapiens | ||
| 4. |  ALA4522598 | 10; FMF-03-198-2 | Activity | 0 | ALA4434179 | Active | Homo sapiens | |||||
| 5. |  ALA4534124 | 36; FMF-03-200-2 | Activity | 0 | ALA4434179 | Active | Homo sapiens | |||||
| 6. |  ALA4563705 | 109; FMF-05-117-1 | IC50 | = | 14 | nM | ALA4434176 | 7.85 | nM | Homo sapiens | ||
| 7. |  ALA4543386 | 108; FMF-05-116-1 | IC50 | = | 332 | nM | ALA4434176 | 6.48 | nM | Homo sapiens | ||
| 8. |  ALA4530961 | 107; FMF-05-027-2 | IC50 | = | 3 | nM | ALA4434176 | 8.52 | nM | Homo sapiens | ||
| 9. |  ALA4451930 | 106; FMF-05-027-1 | IC50 | = | 315 | nM | ALA4434176 | 6.50 | nM | Homo sapiens | ||
| 10. |  ALA4464414 | 105; FMF-05-028-2 | IC50 | = | 221 | nM | ALA4434176 | 6.66 | nM | Homo sapiens | ||
| 11. |  ALA4544087 | 104; FMF-05-028-1 | IC50 | = | 48 | nM | ALA4434176 | 7.32 | nM | Homo sapiens | ||
| 12. |  ALA4467581 | 103; FMF-04-095-1 | IC50 | 0 | ALA4434176 | Not Determined | Homo sapiens | |||||
| 13. |  ALA4566167 | 102; FMF-04-095-1 | IC50 | 0 | ALA4434176 | Not Determined | Homo sapiens | |||||
| 14. | ALA4434727 | 100, 101; FMF-04-159-2 | IC50 | = | 88 | nM | ALA4434176 | 7.06 | nM | Homo sapiens | ||
| 15. |  ALA4474689 | 99; FMF-04-159-1 | IC50 | = | 49 | nM | ALA4434176 | 7.31 | nM | Homo sapiens | ||
| 16. |  ALA4579572 | 98; FMF-04-184-2 | IC50 | = | 6.4 | nM | ALA4434176 | 8.19 | nM | Homo sapiens | ||
| 17. |  ALA4563703 | 97; FMF-04-184-1 | IC50 | = | 0.4 | nM | ALA4434176 | 9.40 | nM | Homo sapiens | ||
| 18. |  ALA4464758 | 96; FMF-05-119-1 | IC50 | = | 50 | nM | ALA4434176 | 7.30 | nM | Homo sapiens | ||
| 19. |  ALA4558269 | 95; FMF-04-097-2 | IC50 | 0 | ALA4434176 | Not Determined | Homo sapiens | |||||
| 20. |  ALA4446451 | 94; FMF-04-097-1 | IC50 | = | 1.6 | nM | ALA4434176 | 8.80 | nM | Homo sapiens |
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