| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4247887 | MB235 | deltaTm | = | 0.7 | degrees C | ALA4234786 | degrees C | Homo sapiens | |||
| 2. |  6-Chlorothiochroman-4-one | MB1200 | deltaTm | = | 1.2 | degrees C | ALA4234786 | degrees C | Homo sapiens | |||
| 3. | ALA4247887 | MB235 | deltaTm | > | 0.5 | degrees C | ALA4234788 | degrees C | Homo sapiens | |||
| 4. | 6-Chlorothiochroman-4-one | MB1200 | deltaTm | > | 0.5 | degrees C | ALA4234788 | degrees C | Homo sapiens | |||
| 5. |  [4-(1H-Pyrrol-1-yl)phenyl]methanol | MB756 | deltaTm | > | 0.5 | degrees C | ALA4234788 | degrees C | Homo sapiens | |||
| 6. |  TBK1 control PROTAC®4 | 4 | IC50 | > | 100 | uM | ALA4219635 | nM | Homo sapiens | |||
| 7. |  ALA4225691 | 6e | IC50 | = | 5.5 | uM | ALA4219635 | 5.26 | nM | Homo sapiens | ||
| 8. |  ALA4226773 | 6d | IC50 | = | 16 | uM | ALA4219635 | 4.80 | nM | Homo sapiens | ||
| 9. |  ALA4227623 | 6c | IC50 | = | 9.9 | uM | ALA4219635 | 5.00 | nM | Homo sapiens | ||
| 10. |  ALA4226398 | 6b | IC50 | = | 25 | uM | ALA4219635 | 4.60 | nM | Homo sapiens | ||
| 11. |  ALA4227365 | 6a | IC50 | > | 100 | uM | ALA4219635 | nM | Homo sapiens | |||
| 12. |  ALA4226250 | 5j | IC50 | = | 800 | nM | ALA4219635 | 6.10 | nM | Homo sapiens | ||
| 13. |  TBK1 PROTAC®3i | 3i | IC50 | = | 4.9 | uM | ALA4219635 | 5.31 | nM | Homo sapiens | ||
| 14. |  ALA3344081 | 7 | IC50 | = | 0.8 | uM | ALA4219635 | 6.10 | nM | Homo sapiens |
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