| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5266174 | SIM 1 | EC50 | = | 0.7 | nM | ALA5249928 | 9.15 | nM | Homo sapiens | ||
| 2. |  ALA5290134 | macroPROTAC-1 | EC50 | = | 25 | nM | ALA5249917 | 7.60 | nM | Homo sapiens | ||
| 3. |  A1874 | 2; A1874 | EC50 | = | 23.1 | nM | ALA5249915 | 7.64 | nM | Homo sapiens | ||
| 4. |  ALA5074720 | 24; AB2 | EC50 | < | 22 | nM | ALA5249914 | nM | Homo sapiens | |||
| 5. |  ARV-771 | 5 | Emax | > | 50 | % | ALA5246323 | % | Homo sapiens | |||
| 6. |  ALA5288732 | 11 | Emax | > | 90 | % | ALA5246323 | % | Homo sapiens | |||
| 7. |  Mz1 | 1; MZ-1 | Emax | > | 90 | % | ALA5246323 | % | Homo sapiens | |||
| 8. | ARV-771 | 5 | DC50 | < | 5 | nM | ALA5246322 | nM | Homo sapiens | |||
| 9. | ALA5288732 | 11 | DC50 | = | 10 | nM | ALA5246322 | nM | Homo sapiens | |||
| 10. | Mz1 | 1; MZ-1 | DC50 | < | 100 | nM | ALA5246322 | nM | Homo sapiens | |||
| 11. | Mz1 | 1; MZ-1 | Emax | > | 90 | % | ALA5246307 | % | Homo sapiens | |||
| 12. | Mz1 | 1; MZ-1 | DC50 | = | 10 | nM | ALA5246306 | nM | Homo sapiens | |||
| 13. | Mz1 | 1; MZ-1 | Activity | = | 90 | % | ALA5246303 | % | Homo sapiens | |||
| 14. |  ALA5279128 | PROTAC 25 | DC50 | < | 1 | nM | ALA5242510 | nM | Homo sapiens | |||
| 15. |  ALA5290390 | 47 | Activity | 0 | ALA5238055 | Not Active | Homo sapiens | |||||
| 16. |  ALA5288300 | 46 | Activity | 0 | ALA5238055 | Not Active | Homo sapiens | |||||
| 17. |  ALA5274328 | 45 | Activity | 0 | ALA5238055 | Not Active | Homo sapiens | |||||
| 18. | Mz1 | 1; MZ-1 | Activity | 0 | ALA5238055 | Active | Homo sapiens | |||||
| 19. |  ALA5284825 | 37 | DC50 | = | 62 | nM | ALA5238051 | nM | Homo sapiens | |||
| 20. |  ALA5291494 | 34 | DC50 | = | 60 | nM | ALA5238051 | nM | Homo sapiens |
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