# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MZP-55 | 10; MZP-55 | Kd | = | 183 | nM | ALA4219529 | 6.74 | nM | Homo sapiens | ||
2. | MZP-54 | 9; MZP-54 | Kd | = | 228 | nM | ALA4219529 | 6.64 | nM | Homo sapiens | ||
3. | ALA4227834 | 8; MZP-61 | Kd | = | 781 | nM | ALA4219529 | 6.11 | nM | Homo sapiens | ||
4. | ALA4227226 | 7; MZ2 | Kd | = | 15 | nM | ALA4219529 | 7.82 | nM | Homo sapiens | ||
5. | Mz1 | 1; MZ-1 | Kd | = | 9 | nM | ALA4219529 | 8.05 | nM | Homo sapiens | ||
6. | ALA4227158 | 5; MZ4 | Kd | = | 26 | nM | ALA4219529 | 7.58 | nM | Homo sapiens | ||
7. | ARV-825 | 6; ARV-825 | Activity | = | 57 | % | ALA4219526 | % | Homo sapiens | |||
8. | MZP-55 | 10; MZP-55 | Activity | = | 47 | % | ALA4219526 | % | Homo sapiens | |||
9. | MZP-54 | 9; MZP-54 | Activity | = | 50 | % | ALA4219526 | % | Homo sapiens | |||
10. | ALA4227834 | 8; MZP-61 | Activity | = | 14 | % | ALA4219526 | % | Homo sapiens | |||
11. | ALA4227226 | 7; MZ2 | Activity | = | 23 | % | ALA4219526 | % | Homo sapiens | |||
12. | Mz1 | 1; MZ-1 | Activity | = | 68 | % | ALA4219526 | % | Homo sapiens | |||
13. | ALA4227158 | 5; MZ4 | Activity | = | 4 | % | ALA4219526 | % | Homo sapiens | |||
14. | GSK1324726A (I-BET726) | 45 | Activity | = | 42 | % | ALA4219526 | % | Homo sapiens | |||
15. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | Activity | = | 20 | % | ALA4219526 | % | Homo sapiens | |||
16. | ARV-825 | 6; ARV-825 | Activity | = | 32 | % | ALA4219525 | % | Homo sapiens | |||
17. | MZP-55 | 10; MZP-55 | Activity | = | 22 | % | ALA4219525 | % | Homo sapiens | |||
18. | MZP-54 | 9; MZP-54 | Activity | = | 28 | % | ALA4219525 | % | Homo sapiens | |||
19. | ALA4227834 | 8; MZP-61 | Activity | = | -156 | % | ALA4219525 | % | Homo sapiens | |||
20. | ALA4227226 | 7; MZ2 | Activity | = | 20 | % | ALA4219525 | % | Homo sapiens |