| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  MZP-55 | 10; MZP-55 | Activity | 0 | ALA4219541 | Not Active | Homo sapiens | |||||
| 2. |  MZP-54 | 9; MZP-54 | Activity | 0 | ALA4219541 | Not Active | Homo sapiens | |||||
| 3. | MZP-55 | 10; MZP-55 | Activity | 0 | ALA4219537 | Not Active | Homo sapiens | |||||
| 4. | MZP-54 | 9; MZP-54 | Activity | 0 | ALA4219537 | Not Active | Homo sapiens | |||||
| 5. |  GSK1324726A (I-BET726) | 45 | Activity | 0 | ALA4219533 | Not Active | Homo sapiens | |||||
| 6. |  (+)-JQ1 (DMSO solution) | (+)-JQ1 | Activity | 0 | ALA4219533 | Not Active | Homo sapiens | |||||
| 7. |  ARV-825 | 6; ARV-825 | Emax | = | 83 | % | ALA4219522 | % | Homo sapiens | |||
| 8. | MZP-55 | 10; MZP-55 | Emax | = | 26 | % | ALA4219522 | % | Homo sapiens | |||
| 9. | MZP-54 | 9; MZP-54 | Emax | = | 43 | % | ALA4219522 | % | Homo sapiens | |||
| 10. |  ALA4227834 | 8; MZP-61 | Emax | = | 37 | % | ALA4219522 | % | Homo sapiens | |||
| 11. |  ALA4227226 | 7; MZ2 | Emax | = | 97 | % | ALA4219522 | % | Homo sapiens | |||
| 12. |  Mz1 | 1; MZ-1 | Emax | = | 98 | % | ALA4219522 | % | Homo sapiens | |||
| 13. |  ALA4227158 | 5; MZ4 | Emax | = | 93 | % | ALA4219522 | % | Homo sapiens | |||
| 14. | ALA4227158 | 5; MZ4 | pDC50 | = | 6.2 | ALA4219516 | Homo sapiens | |||||
| 15. | MZP-55 | 10; MZP-55 | Kd | = | 330 | nM | ALA4219543 | 6.48 | nM | Homo sapiens | ||
| 16. | ARV-825 | 6; ARV-825 | pDC50 | = | 8.2 | ALA4219516 | Homo sapiens | |||||
| 17. | MZP-55 | 10; MZP-55 | Activity | 0 | ALA4219516 | Dose-dependent effect | Homo sapiens | |||||
| 18. | ALA4227226 | 7; MZ2 | Activity | 0 | ALA4219516 | Dose-dependent effect | Homo sapiens | |||||
| 19. | ALA4227226 | 7; MZ2 | pDC50 | = | 6.7 | ALA4219516 | Homo sapiens | |||||
| 20. | Mz1 | 1; MZ-1 | pDC50 | = | 7.4 | ALA4219516 | Homo sapiens |
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