# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5270781 | 38 | IC50 | > | 2 | uM | ALA5252059 | nM | Homo sapiens | |||
2. | ALA5268244 | 51 | IC50 | = | 81 | nM | ALA5243515 | 7.09 | nM | Homo sapiens | ||
3. | ALA5280361 | 50 | IC50 | = | 8.9 | nM | ALA5243515 | 8.05 | nM | Homo sapiens | ||
4. | ALA45177 | 12 (cis) | IC50 | < | 3 | nM | ALA5243513 | nM | Homo sapiens | |||
5. | Ibrutinib (PCI-32765) | SID124898784 | IC50 | = | 200 | nM | ALA5242622 | 6.70 | nM | Homo sapiens | ||
6. | AVL-292 | SPEBRUTINIB | IC50 | = | 4400 | nM | ALA5242622 | 5.36 | nM | Homo sapiens | ||
7. | ALA5285357 | 4; ONO-4059, GS-4059 | IC50 | > | 1 | uM | ALA5242622 | nM | Homo sapiens | |||
8. | ALA5288241 | B2 | INH | < | 50 | % | ALA5238261 | % | Homo sapiens | |||
9. | ALA269538 | 1 | IC50 | > | 250 | uM | ALA5235553 | nM | Homo sapiens | |||
10. | BAY 826 | EUB0000713 | EC50 | = | 7.4 | uM | ALA5213465 | 5.13 | nM | Homo sapiens | ||
11. | ALA4526351 | EUB0000703 | IC50 | = | 7 | uM | ALA5213359 | 5.16 | nM | Homo sapiens | ||
12. | Acalabrutinib (ACP-196) | ACALABRUTINIB | IC50 | > | 10 | uM | ALA5213049 | nM | Homo sapiens | |||
13. | ALA5201686 | 10f | Activity | > | 75 | % | ALA5158083 | % | Homo sapiens | |||
14. | ALA5202420 | 23 | INH | > | 80 | % | ALA5156273 | % | Homo sapiens | |||
15. | ALA4065365 | 6l; E738 | IC50 | = | 10.7 | nM | ALA5151635 | 7.97 | nM | Homo sapiens | ||
16. | ALA5180131 | C13 | Activity | 0 | ALA5136268 | NA | Homo sapiens | |||||
17. | ALA5193966 | 17a | INH | = | 93.9 | % | ALA5135745 | % | Homo sapiens | |||
18. | ALA5179166 | 16a | INH | = | 95 | % | ALA5135745 | % | Homo sapiens | |||
19. | ALA5183704 | 22 | INH | = | 0 | % | ALA5119682 | % | Homo sapiens | |||
20. | ALA3353341 | 16 | INH | = | 20 | % | ALA4430395 | % | Homo sapiens |