# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SKLB-23bb | 23bb | IC50 | = | 31 | nM | ALA5227756 | 7.51 | nM | Homo sapiens | ||
2. | 4-(4-Fluorobenzyl)-8-(1H-pyrrolo[2,3-b]pyridin-5-yl)-3,4-dihydrobenzo[f][1,4]oxazepin-5(2H)-one | 21k | Activity | 0 | ALA5156982 | NA | Homo sapiens | |||||
3. | Paclitaxel | Paclitaxel | TGI | = | 82.9 | % | ALA4425762 | % | Homo sapiens | |||
4. | ALA4538421 | 65 | TGI | = | 85.9 | % | ALA4425761 | % | Homo sapiens | |||
5. | Paclitaxel | Paclitaxel | TGI | = | 85 | % | ALA4425760 | % | Homo sapiens | |||
6. | ALA4538421 | 65 | TGI | = | 88.8 | % | ALA4425760 | % | Homo sapiens | |||
7. | ALA4538421 | 65 | TGI | = | 85.1 | % | ALA4425759 | % | Homo sapiens | |||
8. | ALA4538421 | 65 | TGI | = | 76.5 | % | ALA4425758 | % | Homo sapiens | |||
9. | ALA4538421 | 65 | Activity | 0 | ALA4425744 | Dose-dependent effect | Homo sapiens | |||||
10. | ALA4538421 | 65 | Activity | = | 1.6 | % | ALA4425727 | % | Homo sapiens | |||
11. | ALA4538421 | 65 | Activity | = | 25.5 | % | ALA4425726 | % | Homo sapiens | |||
12. | ALA4538421 | 65 | Activity | = | 40.7 | % | ALA4425725 | % | Homo sapiens | |||
13. | ALA4538421 | 65 | Activity | = | 32.2 | % | ALA4425724 | % | Homo sapiens | |||
14. | ALA4538421 | 65 | Activity | = | 1.3 | % | ALA4425723 | % | Homo sapiens | |||
15. | ALA4538421 | 65 | Activity | = | 22 | % | ALA4425722 | % | Homo sapiens | |||
16. | ALA4538421 | 65 | Activity | = | 42 | % | ALA4425721 | % | Homo sapiens | |||
17. | ALA4538421 | 65 | Activity | = | 34.7 | % | ALA4425720 | % | Homo sapiens | |||
18. | ALA4538421 | 65 | Activity | = | 1.7 | % | ALA4425719 | % | Homo sapiens | |||
19. | ALA4538421 | 65 | Activity | = | 20.9 | % | ALA4425718 | % | Homo sapiens | |||
20. | ALA4538421 | 65 | Activity | = | 37.5 | % | ALA4425717 | % | Homo sapiens |