# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5290046 | 5; HKB99 | EC50 | = | 1.705 | uM | ALA5248667 | 5.77 | nM | Homo sapiens | ||
2. | ALA5290046 | 5; HKB99 | EC50 | = | 1.02 | uM | ALA5248666 | 5.99 | nM | Homo sapiens | ||
3. | ALA301982 | 1 | IC50 | = | 1.3 | uM | ALA5233877 | 5.89 | nM | Homo sapiens | ||
4. | CO-1686 (AVL-301) | ROCILETINIB | IC50 | = | 0.031 | uM | ALA5230872 | 7.51 | nM | Homo sapiens | ||
5. | ALA5283875 | 26 | IC50 | = | 0.65 | uM | ALA5230872 | 6.19 | nM | Homo sapiens | ||
6. | Gefitinib (ZD1839) | Iressa | IC50 | = | 0.006 | uM | ALA5230872 | 8.22 | nM | Homo sapiens | ||
7. | ALA5272742 | 69 | TGI | = | 90 | % | ALA5224330 | % | Homo sapiens | |||
8. | ALA5272742 | 69 | IC50 | = | 6 | nM | ALA5224326 | 8.22 | nM | Homo sapiens | ||
9. | ALA5268128 | 2 | Activity | 0 | ALA5223672 | Active | Homo sapiens | |||||
10. | ALA5290486 | 3 | Activity | 0 | ALA5223668 | Not Active | Homo sapiens | |||||
11. | ALA5268128 | 2 | Activity | = | 51.17 | pg/ml | ALA5223668 | pg/ml | Homo sapiens | |||
12. | ALA5276924 | 1 | Activity | = | 28.2 | pg/ml | ALA5223668 | pg/ml | Homo sapiens | |||
13. | ALA5268128 | 2 | INH | 0 | ALA5223665 | Active | % | Homo sapiens | ||||
14. | ALA5268128 | 2 | Activity | > | 70 | % | ALA5223663 | % | Homo sapiens | |||
15. | ALA5276924 | 1 | Activity | > | 70 | % | ALA5223663 | % | Homo sapiens | |||
16. | ALA5268128 | 2 | Activity | = | 50 | % | ALA5223661 | % | Homo sapiens | |||
17. | ALA5276924 | 1 | Activity | = | 50 | % | ALA5223661 | % | Homo sapiens | |||
18. | ALA5268128 | 2 | Activity | = | 269.14 | % | ALA5223659 | % | Homo sapiens | |||
19. | ALA5276924 | 1 | Activity | = | 23.4 | % | ALA5223659 | % | Homo sapiens | |||
20. | BMS-202 | 1c; BMS-202 | IC50 | = | 8.41 | uM | ALA5223656 | 5.08 | nM | Homo sapiens |