# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5274338 | 2e | IC50 | > | 10 | uM | ALA5251073 | nM | Homo sapiens | |||
2. | Crizotinib | 14, PF-2341066 | IC50 | = | 0.092 | uM | ALA5244683 | 7.04 | nM | Homo sapiens | ||
3. | KRCA 0008 | BDBM193425 | IC50 | = | 0.031 | uM | ALA5244683 | 7.51 | nM | Homo sapiens | ||
4. | ALA5275393 | 9 | IC50 | = | 0.046 | uM | ALA5244683 | 7.34 | nM | Homo sapiens | ||
5. | ALA5182405 | C8 | INH | 0 | ALA5165118 | Active | % | Homo sapiens | ||||
6. | ALA5172782 | I-24 | IC50 | = | 0.027 | uM | ALA5129531 | 7.57 | nM | Homo sapiens | ||
7. | LDK378 | 6, LDK378 | IC50 | = | 0.043 | uM | ALA5129531 | 7.37 | nM | Homo sapiens | ||
8. | ALA5186485 | LB23 | Activity | 0 | ALA5117360 | Active | Homo sapiens | |||||
9. | IPI-504 | 1a | GI50 | = | 76 | nM | ALA4425239 | nM | Homo sapiens | |||
10. | LDK378 | 6, LDK378 | IC50 | = | 27.2 | nM | ALA4388502 | 7.57 | nM | Homo sapiens | ||
11. | ALA4468931 | 15 | IC50 | = | 24.7 | nM | ALA4388502 | 7.61 | nM | Homo sapiens | ||
12. | ALA4542506 | 14 | IC50 | = | 28.5 | nM | ALA4388502 | 7.54 | nM | Homo sapiens | ||
13. | Ceritinib-d7 | 13 | IC50 | = | 28.4 | nM | ALA4388502 | 7.55 | nM | Homo sapiens | ||
14. | ALA4451829 | 12 | IC50 | = | 6 | nM | ALA4388502 | 8.22 | nM | Homo sapiens | ||
15. | ALA4464582 | 11 | IC50 | = | 4 | nM | ALA4388502 | 8.40 | nM | Homo sapiens | ||
16. | JH-VIII-157-02 | 21a | IC50 | = | 5 | nM | ALA4378254 | 8.30 | nM | Homo sapiens | ||
17. | CH5424802 | 18a, CH5424802 | IC50 | = | 9 | nM | ALA4378254 | 8.05 | nM | Homo sapiens | ||
18. | ALA4113131 | ENSARTINIB | Ratio IC50 | = | 10 | ALA4378249 | Homo sapiens | |||||
19. | ALA4113131 | ENSARTINIB | IC50 | = | 15 | nM | ALA4378248 | 7.82 | nM | Homo sapiens | ||
20. | Crizotinib | 14, PF-2341066 | IC50 | = | 180 | nM | ALA4378248 | 6.75 | nM | Homo sapiens |