# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tanshindiol C | 5 | Activity | 0 | ALA3292506 | Active | Homo sapiens | |||||
2. | Tanshindiol C | 5 | Activity | 0 | ALA3292505 | Active | Homo sapiens | |||||
3. | Tanshindiol C | 5 | Activity | 0 | ALA3292504 | Active | Homo sapiens | |||||
4. | Tanshindiol C | 5 | Activity | 0 | ALA3292503 | Active | Homo sapiens | |||||
5. | A 485 | A-485 | Cell Proliferation EC50 | 0.859 | uM | ALA4886688 | uM | Homo sapiens | ||||
6. | Acalabrutinib (ACP-196) | ACALABRUTINIB | IC50 | > | 10 | uM | ALA4841692 | nM | Homo sapiens | |||
7. | ALA4864983 | 26 | IC50 | = | 2.5 | uM | ALA4841692 | 5.60 | nM | Homo sapiens | ||
8. | Tazemetostat (EPZ-6438) | 22, EPZ-6438 | TGI | = | 100 | % | ALA4833707 | % | Homo sapiens | |||
9. | ALA4862681 | 29 | TGI | = | 100 | % | ALA4833707 | % | Homo sapiens | |||
10. | ALA4862681 | 29 | TGI | = | 100 | % | ALA4833706 | % | Homo sapiens | |||
11. | ALA4862681 | 29 | TGI | = | 91.8 | % | ALA4833705 | % | Homo sapiens | |||
12. | Tazemetostat (EPZ-6438) | 22, EPZ-6438 | GI50 | = | 0.002 | uM | ALA4833689 | nM | Homo sapiens | |||
13. | ALA4862681 | 29 | GI50 | = | 0.003 | uM | ALA4833689 | nM | Homo sapiens | |||
14. | ALA4854710 | 9c | Activity | 0 | ALA4827196 | Active | Homo sapiens | |||||
15. | ALA4792256 | 3; GSK126 | TGI | = | 62 | % | ALA4735358 | % | Homo sapiens | |||
16. | A-395 | 2 | TGI | = | 84 | % | ALA4735357 | % | Homo sapiens | |||
17. | A-395 | 2 | IC50 | = | 69 | nM | ALA4735356 | 7.16 | nM | Homo sapiens | ||
18. | ALA4088291 | 19 | EC50 | = | 4.4 | uM | ALA4042642 | 5.36 | nM | Homo sapiens | ||
19. | ALA4101747 | 17 | Activity | 0 | ALA4042642 | Dose-dependent effect | Homo sapiens | |||||
20. | ALA4101747 | 17 | EC50 | = | 3.4 | uM | ALA4042642 | 5.47 | nM | Homo sapiens |