# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2442250 | Bim | Activity | 0 | ALA2445360 | Active | Homo sapiens | |||||
2. | ALA2442251 | Puma | Activity | 0 | ALA2445360 | Active | Homo sapiens | |||||
3. | ALA1916198 | Noxa | Activity | 0 | ALA2445360 | Active | Homo sapiens | |||||
4. | ALA1916195 | Bad | Activity | 0 | ALA2445360 | Active | Homo sapiens | |||||
5. | ALA2442249 | 9 | Activity | 0 | ALA2445116 | Active | Homo sapiens | |||||
6. | 2-methyl-N-[2-({3-[2-(prop-2-enamido)acetamido]phenyl}amino)pyrimidin-5-yl]-5-[3-(trifluoromethyl)benzamido]benzamide | 38 | RatioGI50 | = | 13 | ALA3292716 | Homo sapiens | |||||
7. | 2-methyl-N-(2-{[3-(prop-2-enamido)phenyl]amino}pyrimidin-5-yl)-5-[3-(trifluoromethyl)benzamido]benzamide | 31 | RatioGI50 | = | 13 | ALA3292716 | Homo sapiens | |||||
8. | A 485 | A-485 | Cell Proliferation EC50 | 0.746 | uM | ALA4886684 | uM | Homo sapiens | ||||
9. | ALA2289201 | 5a | INH | 0 | ALA4667793 | Active | % | Homo sapiens | ||||
10. | Tazemetostat (EPZ-6438) | 22, EPZ-6438 | GI50 | = | 1.05 | uM | ALA4833692 | nM | Homo sapiens | |||
11. | ALA4862681 | 29 | GI50 | = | 1.1 | uM | ALA4833692 | nM | Homo sapiens | |||
12. | CAL-101 | 74, GS-1101, CAL-101 | IC50 | = | 0.12 | uM | ALA4728128 | 6.92 | nM | Homo sapiens | ||
13. | ALA4752490 | 8t | IC50 | = | 0.08 | uM | ALA4728128 | 7.10 | nM | Homo sapiens | ||
14. | ALA4788952 | 8s | IC50 | = | 0.1 | uM | ALA4728128 | 7.00 | nM | Homo sapiens | ||
15. | ALA4788725 | 8l | IC50 | = | 0.57 | uM | ALA4728128 | 6.24 | nM | Homo sapiens | ||
16. | ALA4753342 | 8e | IC50 | = | 0.53 | uM | ALA4728128 | 6.28 | nM | Homo sapiens | ||
17. | ALA4750636 | 7f | IC50 | = | 0.18 | uM | ALA4728128 | 6.75 | nM | Homo sapiens | ||
18. | ALA4756563 | 34 | Activity | = | 0.87 | g | ALA4724144 | g | Homo sapiens | |||
19. | CAL-101 | 74, GS-1101, CAL-101 | Activity | = | 1.25 | g | ALA4724144 | g | Homo sapiens | |||
20. | ALA4756563 | 34 | TGI | = | 55.14 | % | ALA4724143 | % | Homo sapiens |