| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5270793 | 93; UM-164 | IC50 | = | 230 | nM | ALA5227289 | 6.64 | nM | Homo sapiens | ||
| 2. |  E6201 | 22, E6201 | IC50 | = | 0.21 | uM | ALA5227193 | 6.68 | nM | Homo sapiens | ||
| 3. |  ALA4448276 | 7 | Activity | 0 | ALA4423502 | Active | Homo sapiens | |||||
| 4. |  ALA4442658 | 2 | Activity | 0 | ALA4423502 | Active | Homo sapiens | |||||
| 5. |  STF 118804 | STF-118804 | Activity | = | 50 | % | ALA4423501 | % | Homo sapiens | |||
| 6. |  ALA4850088 | 612 | T/C | = | -22 | % | ALA4807532 | % | Homo sapiens | |||
| 7. |  Dinaciclib (SCH727965) | DINACICLIB | FC | = | 2.5 | ALA4775160 | Homo sapiens | |||||
| 8. |  ALA2402276 | 1 | INH | 0 | ALA4335577 | Active | % | Homo sapiens | ||||
| 9. |  ALA4217960 | 1 | INH | 0 | ALA4335561 | Active | % | Homo sapiens | ||||
| 10. |  ALA4575227 | 83 | Ratio EC50 | > | 10 | ALA4305075 | Homo sapiens | |||||
| 11. |  ALA4519178 | 81 | Ratio EC50 | > | 10 | ALA4305075 | Homo sapiens | |||||
| 12. |  talazoparib | TALAZOPARIB | EC50 | = | 23.2 | nM | ALA4305074 | 7.63 | nM | Homo sapiens | ||
| 13. | ALA4575227 | 83 | EC50 | > | 50 | uM | ALA4305074 | nM | Homo sapiens | |||
| 14. | ALA4519178 | 81 | EC50 | = | 77.5 | uM | ALA4305074 | 4.11 | nM | Homo sapiens | ||
| 15. |  Olaparib (AZD2281, Ku-0059436) | 47, KU0059436, AZD-2281 | EC50 | = | 7 | uM | ALA4305074 | 5.16 | nM | Homo sapiens | ||
| 16. | talazoparib | TALAZOPARIB | EC50 | = | 1.6 | nM | ALA4305076 | 8.80 | nM | Homo sapiens | ||
| 17. | ALA4575227 | 83 | EC50 | = | 18.68 | uM | ALA4305076 | 4.73 | nM | Homo sapiens | ||
| 18. | ALA4519178 | 81 | EC50 | = | 5.25 | uM | ALA4305076 | 5.28 | nM | Homo sapiens | ||
| 19. | Olaparib (AZD2281, Ku-0059436) | 47, KU0059436, AZD-2281 | EC50 | = | 0.4 | uM | ALA4305076 | 6.40 | nM | Homo sapiens | ||
| 20. |  ALA1276308 | 39 | Activity | 0 | ALA4196360 | Active | Homo sapiens |
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