# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 5-[5-[(3S)-oxolan-3-yl]oxy-6-(1-propan-2-ylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-N-(trideuteriomethyl)pyridine-3-carboxamide | 29 | IC50 | = | 5.5 | nM | ALA5100327 | 8.26 | nM | Mus musculus | ||
2. | ALA5172121 | 28 | IC50 | = | 22 | nM | ALA5100327 | 7.66 | nM | Mus musculus | ||
3. | ALA5203027 | 27 | IC50 | = | 7.2 | nM | ALA5100327 | 8.14 | nM | Mus musculus | ||
4. | ALA5199231 | 26 | IC50 | = | 29 | nM | ALA5100327 | 7.54 | nM | Mus musculus | ||
5. | ALA5174279 | 25 | IC50 | = | 68 | nM | ALA5100327 | 7.17 | nM | Mus musculus | ||
6. | ALA5184953 | 24 | IC50 | = | 13 | nM | ALA5100327 | 7.89 | nM | Mus musculus | ||
7. | ALA5206837 | 23 | IC50 | = | 12 | nM | ALA5100327 | 7.92 | nM | Mus musculus | ||
8. | ALA5187371 | 22 | IC50 | = | 5.4 | nM | ALA5100327 | 8.27 | nM | Mus musculus | ||
9. | ALA5202408 | 21 | IC50 | = | 14 | nM | ALA5100327 | 7.85 | nM | Mus musculus | ||
10. | ALA5208443 | 20 | IC50 | = | 969 | nM | ALA5100327 | 6.01 | nM | Mus musculus | ||
11. | ALA5200643 | 19 | IC50 | = | 15 | nM | ALA5100327 | 7.82 | nM | Mus musculus | ||
12. | ALA5196280 | 17 | IC50 | = | 42 | nM | ALA5100327 | 7.38 | nM | Mus musculus | ||
13. | ALA5202943 | 16 | IC50 | = | 29 | nM | ALA5100327 | 7.54 | nM | Mus musculus | ||
14. | ALA5201556 | 5 | IC50 | = | 33 | nM | ALA5100327 | 7.48 | nM | Mus musculus | ||
15. | ALA5286909 | 19 | IC50 | = | 16 | nM | ALA5258351 | 7.80 | nM | Mus musculus | ||
16. | ALA5290074 | 7 | IC50 | = | 70 | nM | ALA5258351 | 7.16 | nM | Mus musculus | ||
17. | ALA2037208 | 4 | IC50 | = | 6.3 | uM | ALA2038869 | 5.20 | nM | Mus musculus | ||
18. | ALA2037209 | 5 | IC50 | = | 7.7 | uM | ALA2038869 | 5.11 | nM | Mus musculus | ||
19. | ALA2037220 | 16 | IC50 | > | 10 | uM | ALA2038869 | nM | Mus musculus | |||
20. | ALA2037224 | 20 | IC50 | = | 1.7 | uM | ALA2038869 | 5.77 | nM | Mus musculus |