# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4870803 | 43; ARD-2585 | Ratio | = | 30 | ALA4844680 | Homo sapiens | |||||
2. | ALA4870803 | 43; ARD-2585 | TGI | = | 65.9 | % | ALA4844667 | % | Homo sapiens | |||
3. | Enzalutamide | 92 | TGI | = | 45 | % | ALA4844667 | % | Homo sapiens | |||
4. | ALA4870803 | 43; ARD-2585 | TGI | = | 74.3 | % | ALA4844666 | % | Homo sapiens | |||
5. | ALA4870803 | 43; ARD-2585 | TGI | = | 54.9 | % | ALA4844665 | % | Homo sapiens | |||
6. | ALA4870803 | 43; ARD-2585 | INH | = | 78 | % | ALA4844629 | % | Homo sapiens | |||
7. | ALA4854467 | 41 | INH | = | 20 | % | ALA4844629 | % | Homo sapiens | |||
8. | ALA4870803 | 43; ARD-2585 | INH | = | 60 | % | ALA4844628 | % | Homo sapiens | |||
9. | ALA4854467 | 41 | INH | = | 70 | % | ALA4844628 | % | Homo sapiens | |||
10. | ALA4870803 | 43; ARD-2585 | INH | = | 78 | % | ALA4844627 | % | Homo sapiens | |||
11. | ALA4854467 | 41 | INH | = | 74 | % | ALA4844627 | % | Homo sapiens | |||
12. | ALA4872965 | 45 | INH | 0 | ALA4844620 | Active | % | Homo sapiens | ||||
13. | ALA4870803 | 43; ARD-2585 | INH | 0 | ALA4844620 | Active | % | Homo sapiens | ||||
14. | ALA4854467 | 41 | INH | 0 | ALA4844620 | Active | % | Homo sapiens | ||||
15. | ALA4853200 | 48 | IC50 | > | 1000 | nM | ALA4844612 | nM | Homo sapiens | |||
16. | ALA4846811 | 47 | IC50 | > | 1000 | nM | ALA4844612 | nM | Homo sapiens | |||
17. | ALA4873439 | 46 | IC50 | > | 1000 | nM | ALA4844612 | nM | Homo sapiens | |||
18. | ALA4872965 | 45 | IC50 | = | 5.1 | nM | ALA4844612 | 8.29 | nM | Homo sapiens | ||
19. | ALA4849497 | 44 | IC50 | = | 4.3 | nM | ALA4844612 | 8.37 | nM | Homo sapiens | ||
20. | ALA4870803 | 43; ARD-2585 | IC50 | = | 1.5 | nM | ALA4844612 | 8.82 | nM | Homo sapiens |