# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PLX-4720 | PLX-4720 | IC50 | = | 1.5 | uM | ALA5231180 | 5.82 | nM | Homo sapiens | ||
2. | ALA5272340 | 45 | IC50 | = | 1.58 | uM | ALA5231098 | 5.80 | nM | Homo sapiens | ||
3. | ALA5280636 | 14 | IC50 | = | 0.38 | uM | ALA5231089 | 6.42 | nM | Homo sapiens | ||
4. | ALA3805410 | C0B | IC50 | = | 1.75 | uM | ALA5231085 | 5.76 | nM | Homo sapiens | ||
5. | ALA3355898 | 10d | Activity | = | 3.54 | % | ALA3372457 | % | Homo sapiens | |||
6. | ALA3355898 | 10d | Activity | = | 38.25 | % | ALA3372456 | % | Homo sapiens | |||
7. | ALA3355898 | 10d | Activity | = | 47.19 | % | ALA3372455 | % | Homo sapiens | |||
8. | ALA3355898 | 10d | Activity | = | 11.02 | % | ALA3372450 | % | Homo sapiens | |||
9. | ALA3355898 | 10d | Activity | = | 0.09 | % | ALA3372454 | % | Homo sapiens | |||
10. | ALA3355898 | 10d | Activity | = | 17.54 | % | ALA3372453 | % | Homo sapiens | |||
11. | ALA3355898 | 10d | Activity | = | 14.13 | % | ALA3372452 | % | Homo sapiens | |||
12. | ALA3355898 | 10d | Activity | = | 68.24 | % | ALA3372451 | % | Homo sapiens | |||
13. | ALA4167822 | 8b | IC50 | = | 9.2 | uM | ALA4141937 | 5.04 | nM | Homo sapiens | ||
14. | ALA4170805 | 2b | IC50 | = | 7.9 | uM | ALA4141937 | 5.10 | nM | Homo sapiens | ||
15. | ALA4127826 | 25 | GI | 0 | ALA4124365 | Active | Homo sapiens | |||||
16. | Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | GI50 | = | 0.21 | uM | ALA4272242 | nM | Homo sapiens | |||
17. | ALA4286889 | 16 | GI50 | = | 154 | uM | ALA4272242 | nM | Homo sapiens | |||
18. | ALA4294787 | 15 | GI50 | = | 0.42 | uM | ALA4272242 | nM | Homo sapiens | |||
19. | ALA4292278 | 14 | GI50 | = | 70.5 | uM | ALA4272242 | nM | Homo sapiens | |||
20. | ALA4281642 | 13 | GI50 | = | 58.7 | uM | ALA4272242 | nM | Homo sapiens |