# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BPR1R024 | 12; BPRIR024 | IC50 | = | 5.39 | uM | ALA4845045 | 5.27 | nM | |||
2. | Pexidartinib | PEXIDARTINIB | IC50 | > | 10 | uM | ALA4845045 | nM | ||||
3. | BPR1R024 | 12; BPRIR024 | IC50 | = | 0.031 | uM | ALA4845044 | 7.51 | nM | |||
4. | Pexidartinib | PEXIDARTINIB | IC50 | = | 0.056 | uM | ALA4845044 | 7.25 | nM | |||
5. | ALA252913 | 32 | Activity | 0 | ALA4477416 | Active | ||||||
6. | ALA252913 | 32 | Activity | 0 | ALA4477417 | Active | ||||||
7. | ALA2356535 | SID124897877 | Activity | 0 | ALA4425524 | Non-Toxic | ||||||
8. | ALA4476844 | 5 | Activity | 0 | ALA4425522 | Non-Toxic | ||||||
9. | ALA4854616 | 12 | IC50 | = | 40 | uM | ALA4840220 | 4.40 | nM | |||
10. | ALA4869051 | 6f | IC50 | = | 37.3 | uM | ALA4840220 | 4.43 | nM | |||
11. | ALA4853804 | 19 | Activity | < | 7.8 | pg/ml | ALA4836384 | pg/ml | ||||
12. | ALA4859381 | 8 | Activity | < | 7.8 | pg/ml | ALA4836384 | pg/ml | ||||
13. | ALA4853804 | 19 | INH | 0 | ALA4836384 | Dose-Dependent Effect | % | |||||
14. | ALA4859381 | 8 | INH | 0 | ALA4836384 | Dose-Dependent Effect | % | |||||
15. | ALA4865355 | 16 | Activity | < | 7.8 | pg/ml | ALA4836383 | pg/ml | ||||
16. | ALA4864720 | 12 | Activity | < | 7.8 | pg/ml | ALA4836383 | pg/ml | ||||
17. | ALA4873464 | 9 | Activity | < | 7.8 | pg/ml | ALA4836383 | pg/ml | ||||
18. | ALA4867582 | 5 | Activity | < | 7.8 | pg/ml | ALA4836383 | pg/ml | ||||
19. | ALA4865355 | 16 | INH | 0 | ALA4836383 | Dose-Dependent Effect | % | |||||
20. | ALA4864720 | 12 | INH | 0 | ALA4836383 | Dose-Dependent Effect | % |