# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AT13387 | 35 | IC50 | = | 34 | nM | ALA4425253 | 7.47 | nM | Homo sapiens | ||
2. | ALA4448433 | 10a | Activity | = | 59 | % | ALA4386482 | % | Homo sapiens | |||
3. | ALA4448433 | 10a | TGI | 0 | ALA4386483 | Active | Homo sapiens | |||||
4. | Sunitinib | 12b | TGI | 0 | ALA4386543 | Active | Homo sapiens | |||||
5. | Sunitinib | 12b | Activity | 0 | ALA4386542 | Not Active | Homo sapiens | |||||
6. | Imatinib (STI571) | 1 | GI50 | = | 929 | nM | ALA4386530 | nM | Homo sapiens | |||
7. | Sunitinib | 12b | GI50 | = | 47 | nM | ALA4386530 | nM | Homo sapiens | |||
8. | ALA4448433 | 10a | GI50 | = | 1 | nM | ALA4386530 | nM | Homo sapiens | |||
9. | Imatinib (STI571) | 1 | GI50 | = | 929 | nM | ALA4386529 | nM | Homo sapiens | |||
10. | Sunitinib | 12b | GI50 | = | 47 | nM | ALA4386529 | nM | Homo sapiens | |||
11. | ALA4448433 | 10a | GI50 | = | 1 | nM | ALA4386529 | nM | Homo sapiens | |||
12. | ALA4513768 | 15a | Activity | 0 | ALA4379670 | Active | Homo sapiens | |||||
13. | Sunitinib | 12b | Activity | 0 | ALA4379669 | Not Active | Homo sapiens | |||||
14. | ALA4513768 | 15a | Activity | 0 | ALA4379668 | Active | Homo sapiens | |||||
15. | ALA4513768 | 15a | Activity | = | 100 | % | ALA4379667 | % | Homo sapiens | |||
16. | Regorafenib (BAY 73-4506) | 2, BAY-734506 | GI50 | > | 2000 | nM | ALA4379617 | nM | Homo sapiens | |||
17. | Sunitinib | 12b | GI50 | = | 2000 | nM | ALA4379617 | nM | Homo sapiens | |||
18. | Imatinib (STI571) | 1 | GI50 | = | 625 | nM | ALA4379617 | nM | Homo sapiens | |||
19. | ALA4513768 | 15a | GI50 | = | 21 | nM | ALA4379617 | nM | Homo sapiens |