# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Repaglinide | (S)-6al | IC50 | = | 1.25 | uM | ALA4379990 | 5.90 | nM | Rattus norvegicus | ||
2. | ALA4460852 | 5i | IC50 | = | 0.005 | uM | ALA4379990 | 8.32 | nM | Rattus norvegicus | ||
3. | ALA4547171 | 5g | IC50 | = | 0.004 | uM | ALA4379990 | 8.41 | nM | Rattus norvegicus | ||
4. | ALA4529301 | 5c | IC50 | = | 0.002 | uM | ALA4379990 | 8.82 | nM | Rattus norvegicus | ||
5. | ALA4454091 | 5a | IC50 | = | 0.003 | uM | ALA4379990 | 8.55 | nM | Rattus norvegicus | ||
6. | Repaglinide | (S)-6al | INH | = | 99.05 | % | ALA4379991 | % | Rattus norvegicus | |||
7. | Repaglinide | (S)-6al | INH | = | 96.16 | % | ALA4379989 | % | Rattus norvegicus | |||
8. | ALA4460852 | 5i | INH | = | 90.21 | % | ALA4379988 | % | Rattus norvegicus | |||
9. | ALA4547171 | 5g | INH | = | 86.24 | % | ALA4379988 | % | Rattus norvegicus | |||
10. | ALA4529301 | 5c | INH | = | 98.99 | % | ALA4379988 | % | Rattus norvegicus | |||
11. | ALA4454091 | 5a | INH | = | 98.25 | % | ALA4379988 | % | Rattus norvegicus | |||
12. | ALA4460852 | 5i | INH | = | 72.12 | % | ALA4379987 | % | Rattus norvegicus | |||
13. | ALA4547171 | 5g | INH | = | 64.37 | % | ALA4379987 | % | Rattus norvegicus | |||
14. | ALA4529301 | 5c | INH | = | 84.26 | % | ALA4379987 | % | Rattus norvegicus | |||
15. | ALA4454091 | 5a | INH | = | 80.64 | % | ALA4379987 | % | Rattus norvegicus | |||
16. | ALA4529301 | 5c | Activity | 0 | ALA4379980 | Toxic | Rattus norvegicus | |||||
17. | ALA4454091 | 5a | Activity | 0 | ALA4379980 | Toxic | Rattus norvegicus | |||||
18. | ALA4529301 | 5c | Activity | 0 | ALA4379986 | Non-Toxic | Rattus norvegicus | |||||
19. | ALA4454091 | 5a | Activity | 0 | ALA4379986 | Non-Toxic | Rattus norvegicus | |||||
20. | ALA4753376 | 5 | Activity | 0 | ALA4702702 | Active | Rattus norvegicus |