| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  4-(4-Fluorobenzyl)-8-(1H-pyrrolo[2,3-b]pyridin-5-yl)-3,4-dihydrobenzo[f][1,4]oxazepin-5(2H)-one | 21k | Activity | 0 | ALA5156979 | NA | Homo sapiens | |||||
| 2. |  Emavusertib (CA-4948) | 24; CA-4948 | IC50 | = | 1.5 | uM | ALA4673039 | 5.82 | nM | Homo sapiens | ||
| 3. |  ALA4786559 | 59 | IC50 | = | 2.1 | nM | ALA4841295 | 8.68 | nM | Homo sapiens | ||
| 4. |  ALA4876497 | 37 | IC50 | = | 3.2 | nM | ALA4841295 | 8.49 | nM | Homo sapiens | ||
| 5. |  Subasumstat (TAK-981) | TAK-981 | Activity | 0 | ALA4835014 | Active | Homo sapiens | |||||
| 6. |  ALA4856793 | ML-93 | Activity | 0 | ALA4835013 | Active | Homo sapiens | |||||
| 7. | Subasumstat (TAK-981) | TAK-981 | EC50 | = | 0.004 | uM | ALA4835010 | 8.40 | nM | Homo sapiens | ||
| 8. | ALA4856793 | ML-93 | EC50 | = | 0.004 | uM | ALA4835010 | 8.40 | nM | Homo sapiens | ||
| 9. |  ML792 | ML-792 | EC50 | = | 0.055 | uM | ALA4835010 | 7.26 | nM | Homo sapiens | ||
| 10. |  ALA4780218 | 21 | IC50 | = | 10.5 | uM | ALA4767782 | 4.98 | nM | Homo sapiens | ||
| 11. |  ALA4781999 | 18 | IC50 | = | 3.6 | uM | ALA4767782 | 5.44 | nM | Homo sapiens | ||
| 12. |  ALA4778492 | 15 | IC50 | = | 5.8 | uM | ALA4767782 | 5.24 | nM | Homo sapiens | ||
| 13. |  ALA4785023 | 14 | IC50 | = | 2.8 | uM | ALA4767782 | 5.55 | nM | Homo sapiens | ||
| 14. |  ALA4784692 | 11 | IC50 | = | 8.8 | uM | ALA4767782 | 5.06 | nM | Homo sapiens | ||
| 15. |  ALA4787247 | 9 | IC50 | = | 0.8 | uM | ALA4767782 | 6.10 | nM | Homo sapiens | ||
| 16. |  ALA4794821 | 7 | IC50 | = | 3.6 | uM | ALA4767782 | 5.44 | nM | Homo sapiens | ||
| 17. |  ALA4795391 | 6 | IC50 | = | 22.3 | uM | ALA4767782 | 4.65 | nM | Homo sapiens | ||
| 18. |  ALA4799763 | 5-Me | IC50 | 0 | ALA4767782 | Not Determined | Homo sapiens | |||||
| 19. |  ALA4784270 | 4-Me | IC50 | 0 | ALA4767782 | Not Determined | Homo sapiens | |||||
| 20. |  ALA4791581 | 5 | IC50 | = | 0.7 | uM | ALA4767782 | 6.16 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!