# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4515196 | 19a | IC50 | = | 0.47 | uM | ALA4362074 | 6.33 | nM | Homo sapiens | ||
2. | ALA4443725 | 17 | IC50 | = | 0.86 | uM | ALA4362074 | 6.07 | nM | Homo sapiens | ||
3. | EGFR-IN-8 | 1 | Activity | 0 | ALA4363263 | Active | Homo sapiens | |||||
4. | Osimertinib (AZD9291) | 8 | IC50 | = | 0.1 | uM | ALA4363239 | 7.00 | nM | Homo sapiens | ||
5. | Afatinib | BIBW-2992 | IC50 | = | 0.1 | uM | ALA4363239 | 7.00 | nM | Homo sapiens | ||
6. | Erlotinib | Tarceva | IC50 | > | 20 | uM | ALA4363239 | nM | Homo sapiens | |||
7. | Gefitinib (ZD1839) | Iressa | IC50 | = | 10 | uM | ALA4363239 | 5.00 | nM | Homo sapiens | ||
8. | EGFR-IN-8 | 1 | IC50 | = | 0.5 | uM | ALA4363239 | 6.30 | nM | Homo sapiens | ||
9. | EGFR-IN-8 | 1 | IC50 | = | 0.6 | uM | ALA4363234 | 6.22 | nM | Homo sapiens |