# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Imatinib (STI571) | 1 | GI50 | = | 0.058 | uM | ALA4305133 | nM | Homo sapiens | |||
2. | ALA4446361 | 24; CHMFL-KIT-033 | GI50 | = | 0.296 | uM | ALA4305133 | nM | Homo sapiens | |||
3. | (R)-DNMDP | 9; DNMDP | Activity | = | 90 | % | ALA4231518 | % | Homo sapiens | |||
4. | Imatinib (STI571) | 1 | GI50 | = | 0.02 | uM | ALA4012644 | nM | Homo sapiens | |||
5. | ALA4072731 | 31 | GI50 | < | 0.003 | uM | ALA4012644 | nM | Homo sapiens | |||
6. | Imatinib (STI571) | 1 | Activity | 0 | ALA3879110 | Active | Homo sapiens | |||||
7. | Imatinib (STI571) | 1 | Activity | 0 | ALA3879109 | Active | Homo sapiens | |||||
8. | ALA3939150 | 34 | Activity | 0 | ALA3879108 | Active | Homo sapiens | |||||
9. | ALA3939150 | 34 | Activity | 0 | ALA3879107 | Active | Homo sapiens | |||||
10. | Imatinib (STI571) | 1 | GI50 | = | 195 | nM | ALA4386528 | nM | Homo sapiens | |||
11. | Sunitinib | 12b | GI50 | = | 64 | nM | ALA4386528 | nM | Homo sapiens | |||
12. | ALA4448433 | 10a | GI50 | = | 3 | nM | ALA4386528 | nM | Homo sapiens | |||
13. | Imatinib (STI571) | 1 | GI50 | = | 195 | nM | ALA4386526 | nM | Homo sapiens | |||
14. | Sunitinib | 12b | GI50 | = | 64 | nM | ALA4386526 | nM | Homo sapiens | |||
15. | ALA4448433 | 10a | GI50 | = | 3 | nM | ALA4386526 | nM | Homo sapiens | |||
16. | Regorafenib (BAY 73-4506) | 2, BAY-734506 | GI50 | = | 285 | nM | ALA4379615 | nM | Homo sapiens | |||
17. | Sunitinib | 12b | GI50 | = | 64 | nM | ALA4379615 | nM | Homo sapiens | |||
18. | Imatinib (STI571) | 1 | GI50 | = | 195 | nM | ALA4379615 | nM | Homo sapiens | |||
19. | ALA4513768 | 15a | GI50 | = | 5 | nM | ALA4379615 | nM | Homo sapiens | |||
20. | ALA3809935 | 13 | Activity | 0 | ALA3811284 | Active | Homo sapiens |