# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4576024 | 3 | Activity | <= | 99.4 | % | ALA4405118 | % | Homo sapiens | |||
2. | ALA4562996 | 2 | Activity | <= | 99.8 | % | ALA4405118 | % | Homo sapiens | |||
3. | ALA4576024 | 3 | Activity | 0 | ALA4405116 | Active | Homo sapiens | |||||
4. | ALA4562996 | 2 | Activity | 0 | ALA4405116 | Active | Homo sapiens | |||||
5. | ALA4576024 | 3 | Kd | = | 14.34 | uM | ALA4405114 | 4.84 | nM | Homo sapiens | ||
6. | ALA4562996 | 2 | Kd | = | 3.85 | uM | ALA4405114 | 5.42 | nM | Homo sapiens | ||
7. | ALA4438092 | 1 | IC50 | = | 10.4 | uM | ALA4405109 | 4.98 | nM | Homo sapiens | ||
8. | ALA4576024 | 3 | IC50 | = | 3.58 | uM | ALA4405109 | 5.45 | nM | Homo sapiens | ||
9. | ALA4562996 | 2 | IC50 | = | 8.2 | uM | ALA4405109 | 5.09 | nM | Homo sapiens | ||
10. | ALA1813126 | 2a | IC50 | = | 20.1 | uM | ALA4405107 | 4.70 | nM | Homo sapiens | ||
11. | ALA1631706 | 6c | GI50 | = | 5 | uM | ALA4405106 | nM | Homo sapiens | |||
12. | ALA4558745 | 20d; BC-DXI-843 | Activity | 0 | ALA4359580 | Active | Homo sapiens | |||||
13. | ALA4558745 | 20d; BC-DXI-843 | INH | 0 | ALA4359579 | Active | % | Homo sapiens | ||||
14. | ALA4558745 | 20d; BC-DXI-843 | INH | 0 | ALA4359577 | Dose-dependent effect | % | Homo sapiens | ||||
15. | ALA4558745 | 20d; BC-DXI-843 | INH | 0 | ALA4359576 | Active | % | Homo sapiens | ||||
16. | ALA4558745 | 20d; BC-DXI-843 | Activity | 0 | ALA4359575 | Active | Homo sapiens | |||||
17. | ALA4558745 | 20d; BC-DXI-843 | Activity | 0 | ALA4359574 | Not Active | Homo sapiens | |||||
18. | ALA4533418 | 2; BC-DXI-495 | Activity | 0 | ALA4359573 | Not Active | Homo sapiens | |||||
19. | ALA4558745 | 20d; BC-DXI-843 | Activity | 0 | ALA4359573 | Not Active | Homo sapiens | |||||
20. | ALA4558745 | 20d; BC-DXI-843 | Activity | 0 | ALA4359572 | Dose-dependent effect | Homo sapiens |