# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5283010 | 40; TR79 | EC50 | = | 120 | nM | ALA5223588 | 6.92 | nM | Homo sapiens | ||
2. | ALA5275131 | 39; TR57 | EC50 | = | 135 | nM | ALA5223588 | 6.87 | nM | Homo sapiens | ||
3. | ALA5290620 | 37; TR65 | EC50 | = | 120 | nM | ALA5223588 | 6.92 | nM | Homo sapiens | ||
4. | ALA5287429 | 36; TR66 | EC50 | = | 120 | nM | ALA5223588 | 6.92 | nM | Homo sapiens | ||
5. | ALA5290082 | 38; TR27 | EC50 | = | 800 | nM | ALA5223588 | 6.10 | nM | Homo sapiens | ||
6. | TIC10 | DORDAVIPRONE | Activity | 0 | ALA5167803 | Dde | Homo sapiens | |||||
7. | ALA5191392 | 16z | Activity | 0 | ALA5167803 | Dde | Homo sapiens | |||||
8. | ALA5172282 | 16y | Activity | 0 | ALA5167803 | Dde | Homo sapiens | |||||
9. | ALA5205960 | 16x | Activity | 0 | ALA5167803 | Dde | Homo sapiens | |||||
10. | ALA5170508 | 16t | Activity | 0 | ALA5167803 | Dde | Homo sapiens | |||||
11. | ALA5180553 | 16q | Activity | 0 | ALA5167803 | Dde | Homo sapiens | |||||
12. | ALA5191392 | 16z | Ratio | = | 156 | ALA5167718 | Homo sapiens | |||||
13. | TIC10 | DORDAVIPRONE | deltaH | = | -73.87 | kJ/mol | ALA5167717 | kJ/mol | Homo sapiens | |||
14. | ALA5191392 | 16z | deltaH | = | -62.54 | kJ/mol | ALA5167717 | kJ/mol | Homo sapiens | |||
15. | TIC10 | DORDAVIPRONE | deltaS | = | -156.6 | J/mol.K | ALA5167716 | J/mol.K | Homo sapiens | |||
16. | ALA5191392 | 16z | deltaS | = | -77.43 | J/mol.K | ALA5167716 | J/mol.K | Homo sapiens | |||
17. | TIC10 | DORDAVIPRONE | Kd | = | 28.2 | uM | ALA5167715 | 4.55 | nM | Homo sapiens | ||
18. | ALA5191392 | 16z | Kd | = | 0.18 | uM | ALA5167715 | 6.75 | nM | Homo sapiens | ||
19. | ALA5191392 | 16z | Activity | 0 | ALA5167714 | Active | Homo sapiens | |||||
20. | TIC10 | DORDAVIPRONE | Activity | 0 | ALA5167714 | NA | Homo sapiens |