| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  BAY-091 | EUB0001564 | % inhibition | 12.6 | % | ALA4887813 | Not Active | % | Homo sapiens | |||
| 2. |  BAY-885 | BAY-885; 41 | % residual kinase activity | 103 | % | ALA4880999 | Not Active | % | Homo sapiens | |||
| 3. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379185 | nM | Homo sapiens | |||
| 4. |  ALA4459587 | DC-TEADin02 | INH | = | -6 | % | ALA4378922 | % | Homo sapiens | |||
| 5. |  CDK9-IN-7 | 21e | INH | = | 25 | % | ALA4377714 | % | Homo sapiens | |||
| 6. |  ALA4574669 | (R,R)-36n | INH | 0 | ALA4351798 | Not Active | % | Homo sapiens | ||||
| 7. |  ALA4472294 | 11g | Activity | = | 96 | % | ALA4336845 | % | Homo sapiens | |||
| 8. |  ALA4568120 | G28_14 | Activity | = | 58 | % | ALA4335017 | % | Homo sapiens | |||
| 9. |  ALA4455512 | G3_9 | Activity | = | 65 | % | ALA4335017 | % | Homo sapiens | |||
| 10. |  ALA4557538 | 3c; SKLB0533 | Activity | = | 116.5 | % | ALA4314625 | % | Homo sapiens | |||
| 11. |  (1R,3R)-3-[[3-bromo-1-[4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide | 39 | FC | = | 23 | ALA5111604 | Homo sapiens | |||||
| 12. | (1R,3R)-3-[[3-bromo-1-[4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide | 39 | IC50 | = | 118 | nM | ALA5111595 | 6.93 | nM | Homo sapiens | ||
| 13. |  ALA5081774 | EUB0002260 | % inhibition | = | 9 | % | ALA5059071 | Not Active | % | Homo sapiens |
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