# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4534969 | C22 | Activity | 0 | ALA4372627 | Active | Homo sapiens | |||||
2. | NSC 687852 | 2e | INH | 0 | ALA4358853 | Active | % | Homo sapiens | ||||
3. | (R)-2-(2-Chloro-6-fluoro-3-((1-methylpyrrolidin-3-yl)oxy)phenyl)naphtho[2,3-d]oxazole-4,9-dione | 61 | INH | 0 | ALA5112559 | Active | % | Homo sapiens | ||||
4. | ALA5196686 | 35 | INH | 0 | ALA5112559 | Active | % | Homo sapiens | ||||
5. | ALA5180901 | 79 | Activity | 0 | ALA5112558 | Active | Homo sapiens | |||||
6. | ALA5180901 | 79 | Activity | 0 | ALA5112557 | Active | Homo sapiens | |||||
7. | ALA5190411 | 80 | Activity | 0 | ALA5112556 | Active | Homo sapiens | |||||
8. | ALA5180901 | 79 | Activity | 0 | ALA5112555 | Active | Homo sapiens | |||||
9. | (R)-2-(2-Chloro-6-fluoro-3-((1-methylpyrrolidin-3-yl)oxy)phenyl)naphtho[2,3-d]oxazole-4,9-dione | 61 | INH | 0 | ALA5112538 | Active | % | Homo sapiens | ||||
10. | SJB3-019A | SJB3-019A | INH | = | 100 | % | ALA5112532 | % | Homo sapiens | |||
11. | SJB2-043 | 13, SJB2-043 | INH | = | 100 | % | ALA5112532 | % | Homo sapiens | |||
12. | ALA5190411 | 80 | IC50 | = | 6119 | nM | ALA5112525 | 5.21 | nM | Homo sapiens | ||
13. | ALA5180901 | 79 | IC50 | = | 37 | nM | ALA5112525 | 7.43 | nM | Homo sapiens | ||
14. | (R)-2-(2-Chloro-6-fluoro-3-((1-methylpyrrolidin-3-yl)oxy)phenyl)naphtho[2,3-d]oxazole-4,9-dione | 61 | IC50 | = | 0.17 | nM | ALA5112525 | 9.77 | nM | Homo sapiens | ||
15. | ALA5173239 | 60 | IC50 | = | 0.42 | nM | ALA5112525 | 9.38 | nM | Homo sapiens | ||
16. | ALA5196686 | 35 | IC50 | = | 7.1 | nM | ALA5112525 | 8.15 | nM | Homo sapiens | ||
17. | SJB3-019A | SJB3-019A | IC50 | = | 1.7 | nM | ALA5112525 | 8.77 | nM | Homo sapiens | ||
18. | ALA5175998 | 74 | INH | = | 77.2 | % | ALA5112520 | % | Homo sapiens | |||
19. | ALA5175614 | 73 | INH | = | 80.4 | % | ALA5112520 | % | Homo sapiens | |||
20. | ALA5206912 | 72 | INH | = | 77.9 | % | ALA5112520 | % | Homo sapiens |