# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Sunitinib | 12b | INH | 0 | ALA5252775 | Active | % | Homo sapiens | ||||
2. | MnTMPyP pentachloride | 5 | INH | 0 | ALA5252775 | Active | % | Homo sapiens | ||||
3. | ALA3586447 | 11 | INH | = | 0 | % | ALA5252736 | % | Homo sapiens | |||
4. | ALA3586443 | 7 | INH | = | 12 | % | ALA5252736 | % | Homo sapiens | |||
5. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | INH | = | 90 | % | ALA5252736 | % | Homo sapiens | |||
6. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | Kd | > | 10000 | nM | ALA5252715 | nM | Homo sapiens | |||
7. | ALA5274338 | 2e | IC50 | = | 1999 | nM | ALA5251050 | 5.70 | nM | Homo sapiens | ||
8. | ALA5290648 | 2d | IC50 | = | 18.7 | nM | ALA5251033 | 7.73 | nM | Homo sapiens | ||
9. | ALA5274338 | 2e | IC50 | = | 52.6 | nM | ALA5251033 | 7.28 | nM | Homo sapiens | ||
10. | ALA4446835 | 10 | IC50 | = | 150 | nM | ALA5251026 | 6.82 | nM | Homo sapiens | ||
11. | ALA5268244 | 51 | IC50 | = | 1.6 | nM | ALA5243517 | 8.80 | nM | Homo sapiens | ||
12. | ALA5280361 | 50 | IC50 | = | 261 | nM | ALA5243517 | 6.58 | nM | Homo sapiens | ||
13. | ALA5271030 | 7 | IC50 | < | 0.3 | nM | ALA5243462 | nM | Homo sapiens | |||
14. | Futibatinib | BDBM161389 | IC50 | = | 1.6 | nM | ALA5243449 | 8.80 | nM | Homo sapiens | ||
15. | rogaratinib | ROGARATINIB | IC50 | = | 19 | nM | ALA5243440 | 7.72 | nM | Homo sapiens | ||
16. | Erdafitinib (JNJ-42756493) | ERDAFITINIB | IC50 | = | 0.003 | uM | ALA5243064 | 8.52 | nM | Homo sapiens | ||
17. | ALA522892 | 5 | IC50 | = | 9 | nM | ALA5241421 | 8.05 | nM | Homo sapiens | ||
18. | FIIN-3 | 21; FIIN-3 | IC50 | = | 31 | nM | ALA5241411 | 7.51 | nM | Homo sapiens | ||
19. | ALA5269917 | 7; 3D185(HH185) | IC50 | = | 3.6 | nM | ALA5241404 | 8.44 | nM | Homo sapiens | ||
20. | ODM-203 | BDBM247327 | IC50 | = | 6 | nM | ALA5241391 | 8.22 | nM | Homo sapiens |