# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI-3812 | 44 | % Ctrl | = | 98 | % | ALA5304295 | Not Active | % | Homo sapiens | ||
2. | BI-3802 | BI-3802 | % Ctrl | = | 95 | % | ALA5304192 | Not Active | % | Homo sapiens | ||
3. | ALA4639128 | 62 | pIC50 | < | 4.5 | ALA5303915 | nM | Homo sapiens | ||||
4. | GSK620 | 1; 20 | pIC50 | < | 4.5 | ALA5303864 | nM | Homo sapiens | ||||
5. | GSK046 | 15; GSK046 | pIC50 | < | 4.5 | ALA5303815 | nM | Homo sapiens | ||||
6. | ALA3798574 | INK128 | IC50 | = | 230 | nM | ALA3803005 | 6.64 | nM | Homo sapiens | ||
7. | ALA3797834 | 18 | IC50 | = | 77 | nM | ALA3803005 | 7.11 | nM | Homo sapiens | ||
8. | ALA3797933 | 17 | IC50 | = | 5 | nM | ALA3803005 | 8.30 | nM | Homo sapiens | ||
9. | ALA3800138 | 14 | IC50 | = | 99 | nM | ALA3803001 | 7.00 | nM | Homo sapiens | ||
10. | ALA3797590 | 13 | IC50 | = | 302 | nM | ALA3803001 | 6.52 | nM | Homo sapiens | ||
11. | eCF309 | 12 | INH | = | 85 | % | ALA3803012 | % | Homo sapiens | |||
12. | eCF309 | 12 | IC50 | = | 1340 | nM | ALA3803005 | 5.87 | nM | Homo sapiens | ||
13. | eCF309 | 12 | IC50 | = | 1340 | nM | ALA3803001 | 5.87 | nM | Homo sapiens | ||
14. | ALA3799221 | 5 | IC50 | 0 | ALA3803001 | Not Determined | Homo sapiens | |||||
15. | ALA3797750 | 5 | IC50 | = | 0.72 | uM | ALA3802885 | 6.14 | nM | Homo sapiens | ||
16. | ALA3797698 | 7 | IC50 | = | 0.24 | uM | ALA3802885 | 6.62 | nM | Homo sapiens | ||
17. | ALA3797812 | 9 | IC50 | = | 0.14 | uM | ALA3802885 | 6.85 | nM | Homo sapiens | ||
18. | ALA3799511 | 11 | IC50 | = | 0.44 | uM | ALA3802885 | 6.36 | nM | Homo sapiens | ||
19. | ALA3798914 | 13 | IC50 | = | 0.12 | uM | ALA3802885 | 6.92 | nM | Homo sapiens | ||
20. | ALA3799187 | 15 | IC50 | = | 1.9 | uM | ALA3802885 | 5.72 | nM | Homo sapiens |