# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4533471 | H3 | Activity | 0 | ALA4322370 | Not Active | Homo sapiens | |||||
2. | PROTAC Bcl2 degrader-1 | C5 | Activity | 0 | ALA4322368 | Not Active | Homo sapiens | |||||
3. | PROTAC Bcl2 degrader-1 | C5 | Activity | 0 | ALA4322367 | Not Active | Homo sapiens | |||||
4. | PROTAC Bcl2 degrader-1 | C5 | Activity | 0 | ALA4322366 | Not Active | Homo sapiens | |||||
5. | PROTAC Bcl2 degrader-1 | C5 | Activity | 0 | ALA4322343 | Tde | Homo sapiens | |||||
6. | ALA4169380 | 20 | FC | = | 1.3 | ALA4322325 | Homo sapiens | |||||
7. | ALA4169380 | 20 | FC | = | 1.1 | ALA4322324 | Homo sapiens | |||||
8. | PROTAC Bcl2 degrader-1 | C5 | Activity | 0 | ALA4322370 | Dose-dependent effect | Homo sapiens | |||||
9. | ALA4580736 | C5-Me | Activity | 0 | ALA4322362 | Not Active | Homo sapiens | |||||
10. | PROTAC Bcl2 degrader-1 | C5 | DC50 | = | 3 | uM | ALA4322358 | uM | Homo sapiens | |||
11. | ALA4169380 | 20 | FC | = | 1.1 | ALA4322354 | Homo sapiens | |||||
12. | PROTAC Bcl2 degrader-1 | C5 | FC | = | 1 | ALA4322354 | Homo sapiens | |||||
13. | PROTAC Mcl1 degrader-1 | C3 | FC | = | 0.9 | ALA4322354 | Homo sapiens | |||||
14. | ALA4169380 | 20 | FC | = | 1.1 | ALA4322346 | Homo sapiens | |||||
15. | PROTAC Bcl2 degrader-1 | C5 | FC | = | 1 | ALA4322346 | Homo sapiens | |||||
16. | PROTAC Mcl1 degrader-1 | C3 | FC | = | 1 | ALA4322346 | Homo sapiens | |||||
17. | ALA4169380 | 20 | FC | = | 1 | ALA4322353 | Homo sapiens | |||||
18. | PROTAC Bcl2 degrader-1 | C5 | FC | = | 0.7 | ALA4322353 | Homo sapiens | |||||
19. | PROTAC Mcl1 degrader-1 | C3 | FC | = | 1 | ALA4322353 | Homo sapiens | |||||
20. | ALA4530348 | Nap-1 | Activity | 0 | ALA4322374 | Not Active | Homo sapiens |