# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5282858 | AM-A3 | EC50 | = | 1.1 | nM | ALA5249937 | 8.96 | nM | Homo sapiens | ||
2. | ALA4218019 | 3 | Emax | = | 86 | % | ALA5246313 | % | Homo sapiens | |||
3. | ALA4218019 | 3 | DC50 | = | 100 | nM | ALA5246312 | nM | Homo sapiens | |||
4. | ALA5220713 | 62 | DC50 | = | 10 | uM | ALA5217358 | uM | Homo sapiens | |||
5. | ALA5219608 | 61 | DC50 | = | 10 | uM | ALA5217358 | uM | Homo sapiens | |||
6. | ALA4578800 | Ex 140 | Activity | >= | 90 | % | ALA4308526 | % | Homo sapiens | |||
7. | ALA4444805 | Ex 127 | Activity | >= | 90 | % | ALA4308526 | % | Homo sapiens | |||
8. | ALA4577622 | Ex 38; Ex 72 | Activity | >= | 90 | % | ALA4308526 | % | Homo sapiens | |||
9. | ALA4581069 | Ex 25 | Activity | >= | 90 | % | ALA4308526 | % | Homo sapiens | |||
10. | ALA4476831 | Ex 3 | Activity | >= | 90 | % | ALA4308526 | % | Homo sapiens | |||
11. | ALA4578800 | Ex 140 | IC50 | = | 0.6 | nM | ALA4308525 | 9.22 | nM | Homo sapiens | ||
12. | ALA4444805 | Ex 127 | IC50 | = | 0.8 | nM | ALA4308525 | 9.10 | nM | Homo sapiens | ||
13. | ALA4577622 | Ex 38; Ex 72 | IC50 | = | 0.3 | nM | ALA4308525 | 9.52 | nM | Homo sapiens | ||
14. | ALA4581069 | Ex 25 | IC50 | = | 0.4 | nM | ALA4308525 | 9.40 | nM | Homo sapiens | ||
15. | ALA4476831 | Ex 3 | IC50 | = | 0.3 | nM | ALA4308525 | 9.52 | nM | Homo sapiens | ||
16. | Fulvestrant | 3, ICI-182780 | Activity | = | 100 | % | ALA4308526 | % | Homo sapiens | |||
17. | ALA4750940 | VH032-PERM3-R7 | Activity | = | 84 | % | ALA4726657 | % | Homo sapiens | |||
18. | ALA4750940 | VH032-PERM3-R7 | Activity | = | 108 | % | ALA4726642 | % | Homo sapiens | |||
19. | ALA4750940 | VH032-PERM3-R7 | Activity | = | 92 | % | ALA4726639 | % | Homo sapiens | |||
20. | ALA4750940 | VH032-PERM3-R7 | Activity | = | 57 | % | ALA4726610 | % | Homo sapiens |