# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Halopemide | 1, halopemide | IC50 | = | 300 | nM | ALA4329646 | 6.52 | nM | Homo sapiens | ||
2. | (1R,2R)-N-([S]-1-{4-[5-bromo-2-oxo-2,3-dihydro-1H-benzo(d)imidazol-1-yl]piperidin-1-yl}propan-2-yl)-2-phenylcyclopropanecarboxamide | 13o | IC50 | = | 6400 | nM | ALA4329646 | 5.19 | nM | Homo sapiens | ||
3. | VU0364739 | 22a | IC50 | = | 20 | nM | ALA4329646 | 7.70 | nM | Homo sapiens | ||
4. | ML298 | 7g, ML298, CID53393915 | IC50 | = | 355 | nM | ALA4329646 | 6.45 | nM | Homo sapiens | ||
5. | ML299 | 5; ML299 | IC50 | = | 20 | nM | ALA4329646 | 7.70 | nM | Homo sapiens | ||
6. | ALA3580438 | 6; ML395 | IC50 | = | 360 | nM | ALA4329646 | 6.44 | nM | Homo sapiens | ||
7. | ALA4515874 | (S)-14a | IC50 | = | 70 | nM | ALA4329650 | 7.16 | nM | Homo sapiens | ||
8. | ALA4584012 | (R)-14a | IC50 | = | 810 | nM | ALA4329650 | 6.09 | nM | Homo sapiens | ||
9. | ALA4514153 | (S)-16a | IC50 | = | 150 | nM | ALA4329650 | 6.82 | nM | Homo sapiens | ||
10. | ALA4591820 | (R)-16a | IC50 | = | 4000 | nM | ALA4329650 | 5.40 | nM | Homo sapiens | ||
11. | ALA4475943 | (S)-14b | IC50 | = | 2.5 | nM | ALA4329650 | 8.60 | nM | Homo sapiens | ||
12. | ALA4436548 | (R)-14b | IC50 | = | 43 | nM | ALA4329650 | 7.37 | nM | Homo sapiens | ||
13. | ALA4453586 | (S)-16b | IC50 | = | 12 | nM | ALA4329650 | 7.92 | nM | Homo sapiens | ||
14. | ALA4448918 | (R)-16b | IC50 | = | 140 | nM | ALA4329650 | 6.85 | nM | Homo sapiens | ||
15. | ALA3923136 | (S)-14c | IC50 | = | 60 | nM | ALA4329650 | 7.22 | nM | Homo sapiens | ||
16. | ALA4109224 | BDBM179741 | IC50 | = | 450 | nM | ALA4329650 | 6.35 | nM | Homo sapiens | ||
17. | ALA4570440 | (S)-16c | IC50 | = | 115 | nM | ALA4329650 | 6.94 | nM | Homo sapiens | ||
18. | ALA3902347 | BDBM179736 | IC50 | = | 700 | nM | ALA4329650 | 6.16 | nM | Homo sapiens | ||
19. | ALA3983405 | (S)-14d | IC50 | = | 220 | nM | ALA4329650 | 6.66 | nM | Homo sapiens | ||
20. | ALA4109788 | BDBM179738 | IC50 | = | 3175 | nM | ALA4329650 | 5.50 | nM | Homo sapiens |