# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI-3812 | 44 | % Ctrl | = | 99 | % | ALA5304297 | Not Active | % | Homo sapiens | ||
2. | BI-3802 | BI-3802 | % Ctrl | = | 91 | % | ALA5304194 | Not Active | % | Homo sapiens | ||
3. | LX7101 | 28, LX7101 | INH | > | 90 | % | ALA3801316 | % | Homo sapiens | |||
4. | ALA3797874 | 3 | IC50 | > | 1000 | nM | ALA3801113 | nM | Homo sapiens | |||
5. | ALA3799326 | 2 | IC50 | > | 1000 | nM | ALA3801113 | nM | Homo sapiens | |||
6. | LX7101 | 28, LX7101 | IC50 | < | 1 | nM | ALA3801113 | nM | Homo sapiens | |||
7. | ALA3792850 | 26 | INH | = | -1.4 | % | ALA3794947 | % | Homo sapiens | |||
8. | ALA3793843 | 24 | INH | = | 2.7 | % | ALA3794947 | % | Homo sapiens | |||
9. | ALA508964 | 13 | INH | = | 3.1 | % | ALA3794947 | % | Homo sapiens | |||
10. | ALA3785951 | 33 | IC50 | > | 10 | uM | ALA3790303 | nM | Homo sapiens | |||
11. | ALA3786167 | 28 | IC50 | > | 10 | uM | ALA3790303 | nM | Homo sapiens | |||
12. | ALA3785500 | 3 | IC50 | > | 10 | uM | ALA3790303 | nM | Homo sapiens | |||
13. | ALA3787112 | 2 | IC50 | = | 0.78 | uM | ALA3790303 | 6.11 | nM | Homo sapiens | ||
14. | ALA3787614 | 17 | IC50 | > | 10 | uM | ALA3790303 | nM | Homo sapiens | |||
15. | ALA1614712 | 1; NVP-AEW541 | IC50 | > | 10 | uM | ALA3790303 | nM | Homo sapiens | |||
16. | ALA3780032 | 5; IACS-4759 | INH | 0 | ALA3782386 | Not Active | % | Homo sapiens | ||||
17. | ALA3774448 | 17 | INH | 0 | ALA3776511 | Not Active | % | Homo sapiens | ||||
18. | ALA3775393 | 16 | INH | 0 | ALA3776510 | Not Active | % | Homo sapiens | ||||
19. | ALA3771285 | 12 | Activity | = | 94 | % | ALA3771946 | % | Homo sapiens | |||
20. | Erlotinib | Tarceva | INH | = | -10 | % | ALA3761597 | % | Homo sapiens |