# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405516 | % | Homo sapiens | |||
2. | ALA4794578 | 7 | Activity | = | 110.23 | % | ALA4721500 | % | Homo sapiens | |||
3. | ALA4750196 | 6g | Activity | = | 96.23 | % | ALA4720942 | % | Homo sapiens | |||
4. | Staurosporine | 1 (Staurosporine) | IC50 | = | 1.29 | 10^-9M | ALA4720597 | 8.89 | nM | Homo sapiens | ||
5. | GSK'963 | 9 | INH | 0 | ALA4352499 | Active | % | Homo sapiens | ||||
6. | Staurosporine | 1 (Staurosporine) | IC50 | = | 6.8 | 10'-9M | ALA4328560 | 8.17 | nM | Homo sapiens | ||
7. | Staurosporine | 1 (Staurosporine) | Activity | < | 65 | % | ALA4328196 | % | Homo sapiens | |||
8. | ALA4446405 | 7b; ASR352 | Activity | = | 104.7 | % | ALA4327832 | % | Homo sapiens | |||
9. | ALA4438024 | 7a; NSC30049; NSC49L | Activity | = | 97.99 | % | ALA4327832 | % | Homo sapiens | |||
10. | ALA4576489 | 8b | Kd | = | 154 | nM | ALA4322837 | 6.81 | nM | Homo sapiens | ||
11. | ALA4465866 | 8a | Kd | = | 148 | nM | ALA4322837 | 6.83 | nM | Homo sapiens | ||
12. | ALA4749141 | 44 | Activity | = | 101.08 | % | ALA4674242 | % | Homo sapiens | |||
13. | ALA4785602 | 46 | Activity | = | 106.32 | % | ALA4674242 | % | Homo sapiens | |||
14. | BI 605906 | BI605906 | % Ctrl | 103 | % | ALA4887315 | Not Active | % | Homo sapiens | |||
15. | ALA4097778 | 16h | pIC50 | 6 | ALA4885400 | nM | Homo sapiens | |||||
16. | ALA4549667 | EUB0000720 | pIC50 | 6 | ALA4885114 | nM | Homo sapiens | |||||
17. | ALA4088216 | 14 | pIC50 | 6 | ALA4884823 | nM | Homo sapiens | |||||
18. | ALA4634455 | 3a; TRC-2885 | INH | = | 50 | % | ALA4606503 | % | Homo sapiens | |||
19. | Alisertib (MLN8237) | 9, MLN-8237 | Kd apparent | > | 30000 | nM | ALA3991838 | Inactive | nM | Homo sapiens | ||
20. | LGX 818 | ENCORAFENIB | Kd apparent | > | 30000 | nM | ALA3991838 | Inactive | nM | Homo sapiens |