# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1221574 | 21, P49-F6 | INH | 0 | ALA4421970 | Active | % | Homo sapiens | ||||
2. | ALA1221574 | 21, P49-F6 | Ki | = | 1.36 | uM | ALA4421969 | 5.87 | nM | Homo sapiens | ||
3. | ALA1221574 | 21, P49-F6 | INH | 0 | ALA4421968 | Active | % | Homo sapiens | ||||
4. | ALA1221574 | 21, P49-F6 | INH | 0 | ALA4421965 | Active | % | Homo sapiens | ||||
5. | ALA4567250 | P61-A6; P61-B7 | INH | 0 | ALA4421949 | Not Active | % | Homo sapiens | ||||
6. | ALA1221574 | 21, P49-F6 | INH | 0 | ALA4421948 | Active | % | Homo sapiens | ||||
7. | ALA4567250 | P61-A6; P61-B7 | INH | 0 | ALA4421947 | Not Active | % | Homo sapiens | ||||
8. | ALA4439180 | P5-H6; A03C40; UC22 | INH | 0 | ALA4421939 | Active | % | Homo sapiens | ||||
9. | ALA1366797 | SID56463724 | INH | 0 | ALA4421940 | Not Active | % | Homo sapiens | ||||
10. | ALA4558573 | Fig 29B, R4C2; Table 3, R11C2; P8-H6 | IC50 | = | 3.1 | uM | ALA4421918 | 5.51 | nM | Homo sapiens | ||
11. | ALA4467525 | Fig 29B, R5C2; Table 3, R12C2; P8-H7 | IC50 | = | 7 | uM | ALA4421918 | 5.16 | nM | Homo sapiens | ||
12. | ALA4443727 | Fig 29C, R3C2; P8-G7; Table 3, R17C2 | IC50 | = | 4.7 | uM | ALA4421918 | 5.33 | nM | Homo sapiens | ||
13. | ALA4469845 | P49-F5 | IC50 | = | 7 | uM | ALA4421918 | 5.16 | nM | Homo sapiens | ||
14. | ALA1221621 | 23, P23-D6 | IC50 | = | 4.5 | uM | ALA4421918 | 5.35 | nM | Homo sapiens | ||
15. | ALA4518286 | P47-D11 | IC50 | = | 3.6 | uM | ALA4421918 | 5.44 | nM | Homo sapiens | ||
16. | ALA4456846 | P49-A6 | IC50 | = | 4.8 | uM | ALA4421918 | 5.32 | nM | Homo sapiens | ||
17. | ALA1221574 | 21, P49-F6 | IC50 | = | 2.1 | uM | ALA4421918 | 5.68 | nM | Homo sapiens | ||
18. | ALA1221575 | 22, P50-E11 | IC50 | = | 2.2 | uM | ALA4421918 | 5.66 | nM | Homo sapiens | ||
19. | ALA4438314 | 13 | LED | = | 1 | mM | ALA4315908 | mM | Homo sapiens | |||
20. | ALA4514446 | 14 | LED | = | 5 | mM | ALA4315908 | mM | Homo sapiens |