# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5285300 | 24 | INH | = | 93 | % | ALA5236442 | % | Homo sapiens | |||
2. | ALA5094892 | S9 | INH | = | 69.8 | % | ALA5236442 | % | Homo sapiens | |||
3. | Pep 2-8 | Pep2-8 | INH | = | 36.5 | % | ALA5236442 | % | Homo sapiens | |||
4. | ALA5271747 | 40 | Emax | = | 38 | % | ALA5236438 | % | Homo sapiens | |||
5. | ALA5278292 | 41; 13PCSK9i | Emax | = | 77 | % | ALA5236438 | % | Homo sapiens | |||
6. | ALA5271747 | 40 | EC50 | = | 0.106 | uM | ALA5236437 | 6.97 | nM | Homo sapiens | ||
7. | ALA4228379 | Ref 37, cpd 7 | EC50 | = | 6 | uM | ALA5236437 | 5.22 | nM | Homo sapiens | ||
8. | ALA5278292 | 41; 13PCSK9i | EC50 | = | 0.17 | uM | ALA5236437 | 6.77 | nM | Homo sapiens | ||
9. | ALA5278292 | 41; 13PCSK9i | Emax | = | 90 | % | ALA5236436 | % | Homo sapiens | |||
10. | ALA5278854 | 19; P5-Best | INH | = | 254 | % | ALA5236428 | % | Homo sapiens | |||
11. | ALA5277547 | 18; P5-met | INH | = | 104 | % | ALA5236428 | % | Homo sapiens | |||
12. | ALA5287357 | 17; P5 | INH | = | 100 | % | ALA5236428 | % | Homo sapiens | |||
13. | ALA5278854 | 19; P5-Best | INH | = | 156 | % | ALA5236427 | % | Homo sapiens | |||
14. | ALA5277547 | 18; P5-met | INH | = | 90 | % | ALA5236427 | % | Homo sapiens | |||
15. | ALA5287357 | 17; P5 | INH | = | 99 | % | ALA5236427 | % | Homo sapiens | |||
16. | ALA4472590 | T9 | INH | = | 102.3 | % | ALA5236426 | % | Homo sapiens | |||
17. | ALA4472590 | T9 | INH | = | 74 | % | ALA5236425 | % | Homo sapiens | |||
18. | ALA4228379 | Ref 37, cpd 7 | IC50 | = | 11.2 | uM | ALA5236424 | 4.95 | nM | Homo sapiens | ||
19. | ALA5278292 | 41; 13PCSK9i | IC50 | = | 0.002 | uM | ALA5236424 | 8.70 | nM | Homo sapiens | ||
20. | ALA5285300 | 24 | IC50 | = | 14.5 | uM | ALA5236424 | 4.84 | nM | Homo sapiens |