# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF 04418948 | 15, PF-04418948 | % inhibition | -3 | % | ALA4887016 | Not Active | % | Homo sapiens | |||
2. | ABT 724 | 3a | % inhibition | 51 | % | ALA4880355 | Not Active | % | Homo sapiens | |||
3. | ABT-100 | EUB0000289 | % inhibition | 50 | % | ALA4880194 | Not Active | % | Homo sapiens | |||
4. | ALA4875978 | ML-SI1; racemic mixture(55:45) | IC50 | = | 15 | uM | ALA4819516 | 4.82 | nM | Homo sapiens | ||
5. | ALA4856175 | (+/-)-trans-ML-SI3 | IC50 | = | 2.6 | uM | ALA4819516 | 5.58 | nM | Homo sapiens | ||
6. | ALA4875978 | ML-SI1; racemic mixture(55:45) | INH | 0 | ALA4819515 | Not Active | % | Homo sapiens | ||||
7. | ALA4856175 | (+/-)-trans-ML-SI3 | INH | 0 | ALA4819515 | Active | % | Homo sapiens | ||||
8. | ALA4875551 | 31 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
9. | ALA4851134 | 28 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
10. | ALA4874310 | 27 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
11. | ALA4855589 | 26 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
12. | ALA4856325 | 25 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
13. | ALA4870275 | 23 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
14. | ALA4855846 | 22 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
15. | ALA4849322 | 21 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
16. | ALA4858349 | 20 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
17. | ALA4847300 | 18 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
18. | ALA4857820 | 17 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
19. | (1R,2R)-ML-SI3 | (+)-trans-ML-SI3 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens | |||||
20. | ALA4856175 | (+/-)-trans-ML-SI3 | EC50 | 0 | ALA4819511 | Not Active | Homo sapiens |