# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AMG-517 | 23 | IC50 | = | 0.9 | nM | ALA5247267 | 9.05 | nM | Rattus norvegicus | ||
2. | ALA229431 | 12 | IC50 | = | 27 | nM | ALA5247267 | 7.57 | nM | Rattus norvegicus | ||
3. | ALA375460 | 13 | IC50 | = | 350 | nM | ALA5247267 | 6.46 | nM | Rattus norvegicus | ||
4. | ALA229432 | 14 | IC50 | = | 330 | nM | ALA5247267 | 6.48 | nM | Rattus norvegicus | ||
5. | ALA227209 | 16e | IC50 | = | 380 | nM | ALA5247267 | 6.42 | nM | Rattus norvegicus | ||
6. | AMG628 | 16p, AMG-628 | IC50 | = | 3.7 | nM | ALA5247267 | 8.43 | nM | Rattus norvegicus | ||
7. | Capsaicin | 1 (capsaicin) | Activity | 0 | ALA4379545 | Active | Rattus norvegicus | |||||
8. | MDR-652 | 4; MDR-652 | Activity | 0 | ALA4379543 | Active | Rattus norvegicus | |||||
9. | MDR-652 | 4; MDR-652 | Activity | = | 50 | % | ALA4379542 | % | Rattus norvegicus | |||
10. | MDR-652 | 4; MDR-652 | Ratio Ki | = | 80 | ALA4379514 | Rattus norvegicus | |||||
11. | Capsaicin | 1 (capsaicin) | EC50 | = | 44.8 | nM | ALA4379512 | 7.35 | nM | Rattus norvegicus | ||
12. | MDR-652 | 4; MDR-652 | EC50 | = | 93 | nM | ALA4379512 | 7.03 | nM | Rattus norvegicus | ||
13. | Capsaicin | 1 (capsaicin) | Ki | = | 1810 | nM | ALA4379511 | 5.74 | nM | Rattus norvegicus | ||
14. | MDR-652 | 4; MDR-652 | Ki | = | 23.8 | nM | ALA4379511 | 7.62 | nM | Rattus norvegicus | ||
15. | Clemizole | SID11110952 | IC50 | > | 20 | uM | ALA4377084 | nM | Rattus norvegicus | |||
16. | ALA4778235 | 4aa | pEC50 | = | 6.8 | ALA4734809 | 6.80 | nM | Rattus norvegicus | |||
17. | ALA472897 | 1 | pEC50 | = | 6.4 | ALA4734809 | 6.40 | nM | Rattus norvegicus | |||
18. | ALA4747170 | 2aa | pEC50 | = | 7.2 | ALA4734809 | 7.20 | nM | Rattus norvegicus | |||
19. | ALA472898 | 3 | pEC50 | = | 7.8 | ALA4734809 | 7.80 | nM | Rattus norvegicus | |||
20. | Arvanil | 1d | pEC50 | 0 | ALA4734809 | Not Determined | Rattus norvegicus |