# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4081807 | 28c | Activity | 0 | ALA3998987 | Active | Homo sapiens | |||||
2. | ALA4081807 | 28c | Activity | 0 | ALA3998985 | Dose-dependent effect | Homo sapiens | |||||
3. | ALA4081807 | 28c | Activity | = | 27 | % | ALA3998984 | % | Homo sapiens | |||
4. | Tamoxifen | Tamoxifen | Activity | 0 | ALA3998983 | Not Active | Homo sapiens | |||||
5. | ALA4081807 | 28c | Activity | = | 49 | % | ALA3998983 | % | Homo sapiens | |||
6. | ALA4070169 | 28a | Activity | = | 26.7 | % | ALA3998983 | % | Homo sapiens | |||
7. | Brilanestrant (GDC-0810) | BRILANESTRANT | Activity | = | 21 | % | ALA3998983 | % | Homo sapiens | |||
8. | ALA4081807 | 28c | GI | 0 | ALA3998981 | Active | Homo sapiens | |||||
9. | ALA4081807 | 28c | GI | 0 | ALA3998980 | Active | Homo sapiens | |||||
10. | Brilanestrant (GDC-0810) | BRILANESTRANT | GI | 0 | ALA3998980 | Active | Homo sapiens | |||||
11. | Fulvestrant | 3, ICI-182780 | Activity | 0 | ALA4356709 | Active | Homo sapiens | |||||
12. | Tamoxifen | Tamoxifen | Activity | 0 | ALA4356708 | Not Active | Homo sapiens | |||||
13. | ALA4533964 | 37d | Activity | 0 | ALA4356708 | Active | Homo sapiens | |||||
14. | ALA4533964 | 37d | Activity | 0 | ALA4356698 | Active | Homo sapiens | |||||
15. | ALA4543096 | 30f | Activity | 0 | ALA4356698 | Active | Homo sapiens | |||||
16. | Fulvestrant | 3, ICI-182780 | Activity | 0 | ALA4356698 | Active | Homo sapiens | |||||
17. | ALA4475977 | 220b | IC50 | = | 4 | uM | ALA4324448 | 5.40 | nM | Homo sapiens | ||
18. | ALA4443331 | 220c | IC50 | = | 4 | uM | ALA4324448 | 5.40 | nM | Homo sapiens | ||
19. | ALA4637258 | 27.HCl | TGI | 0 | ALA4612593 | Active | Homo sapiens | |||||
20. | ALA4637258 | 27.HCl | TGI | = | 106 | % | ALA4612589 | % | Homo sapiens |